SCHEMBL14229016

SCHEMBL14229016

CCCCN(C(=O)CCC)c1ccccc1C

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.68
ALDH1A1 P00352 1/20 0.68
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
POLB P06746 1/20 0.48
CYP3A4 P08684 2/20 0.47
LMNA P02545 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.47
NPC1 O15118 1/20 0.42
JAK2 O60674 1/20 0.42
RAB9A P51151 1/20 0.42
PAX8 Q06710 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
OPRM1 P35372 1/20 0.42
TSHR P16473 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
MLYCD O95822 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4158666 0.91 TP53 (0.60) TP53ALDH1A1MEN1KMT2APOLB
SCHEMBL4158674 0.88 TP53 (0.56) TP53ALDH1A1MEN1KMT2APOLB
SCHEMBL4157179 0.87 TP53 (0.63) TP53ALDH1A1MEN1KMT2APOLB
SCHEMBL4055701 0.85 CYP3A4 (0.58) TP53ALDH1A1MEN1KMT2APOLB
SCHEMBL11446155 0.84 ALDH1A1 (0.62) TP53ALDH1A1MEN1KMT2APOLB
SCHEMBL14200322 0.84 TP53 (0.63) TP53ALDH1A1MEN1KMT2APOLB
SCHEMBL14229096 0.83 TP53 (0.51) TP53ALDH1A1CYP3A4NPC1JAK2
SCHEMBL14229099 0.83 TP53 (0.51) TP53ALDH1A1CYP3A4LMNANPC1
SCHEMBL4058268 0.83 POLB (0.59) TP53ALDH1A1MEN1KMT2APOLB
SCHEMBL14229516 0.82 TP53 (0.50) TP53ALDH1A1KMT2ALMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed