SCHEMBL14200322

SCHEMBL14200322

CCCCN(C(=O)CC(C)(C)C)c1ccccc1C

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.63
ALDH1A1 P00352 3/20 0.63
CYP3A4 P08684 3/20 0.43
LMNA P02545 2/20 0.43
TRPM8 Q7Z2W7 1/20 0.43
POLB P06746 1/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PAX8 Q06710 2/20 0.40
JAK2 O60674 1/20 0.40
TSHR P16473 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MLYCD O95822 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200331 0.84 TP53 (0.48) TP53ALDH1A1LMNANPC1RAB9A
SCHEMBL14200334 0.84 TP53 (0.45) TP53ALDH1A1LMNAPOLBNPC1
SCHEMBL14229016 0.84 TP53 (0.68) TP53ALDH1A1CYP3A4LMNATRPM8
SCHEMBL14200351 0.82 SIGMAR1 (0.44) TP53ALDH1A1LMNANPC1RAB9A
SCHEMBL14200339 0.82 CYP1A2 (0.48) TP53ALDH1A1CYP3A4POLBNPC1
SCHEMBL14200236 0.81 NPC1 (0.60) TP53ALDH1A1CYP3A4TRPM8NPC1
SCHEMBL11446155 0.80 ALDH1A1 (0.62) TP53ALDH1A1CYP3A4LMNATRPM8
SCHEMBL28038835 0.79 TP53 (0.54) TP53ALDH1A1CYP3A4LMNATRPM8
SCHEMBL14200327 0.78 NPC1 (0.46) TP53ALDH1A1CYP3A4NPC1RAB9A
SCHEMBL30375032 0.78 TP53 (0.59) TP53ALDH1A1CYP3A4LMNATRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed