SCHEMBL14200852

SCHEMBL14200852

CCCN(Cc1ccc(F)c(F)c1)C(=O)CC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.51
POLB P06746 1/20 0.44
APEX1 P27695 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HTT P42858 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MITF O75030 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SOAT1 P35610 1/20 0.39
HDAC1 Q13547 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
MLYCD O95822 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200903 0.92 RIPK1 (0.49) RIPK1HTTALDH1A1KDM4EMITF
SCHEMBL14229280 0.85 RIPK1 (0.48) RIPK1POLBAPEX1TDP1HTT
SCHEMBL14200898 0.82 HDAC1 (0.40) POLBAPEX1TDP1HDAC1HDAC6
SCHEMBL14200786 0.81 TSHR (0.41) POLBAPEX1TDP1ALDH1A1HDAC1
SCHEMBL14200735 0.79 APP (0.47) HTTALDH1A1KDM4EMITFNPSR1
SCHEMBL14200919 0.78 GRIN2D (0.46) POLBAPEX1TDP1HTTALDH1A1
SCHEMBL14200864 0.78 RIPK1 (0.48) RIPK1HTTALDH1A1KDM4EMITF
SCHEMBL14200851 0.77 RIPK1 (0.50) RIPK1HTTALDH1A1KDM4EMITF
SCHEMBL14200878 0.77 RIPK1 (0.47) RIPK1HTTALDH1A1KDM4EMITF
SCHEMBL14229063 0.77 HDAC1 (0.53) RIPK1HTTALDH1A1KDM4EMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed