SCHEMBL14229265

SCHEMBL14229265

CCCC(=O)N(c1ccc(F)c(Br)c1)C(C)CC

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TP53 P04637 1/20 0.33
KDM4E B2RXH2 2/20 0.33
IDO1 P14902 5/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
ABCC9 O60706 1/20 0.30
ABCC8 Q09428 1/20 0.30
KCNJ11 Q14654 1/20 0.30
KCNJ8 Q15842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229455 0.91 CYP1A2 (0.35) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL14229460 0.89 NPSR1 (0.37) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL14229738 0.88 CYP1A2 (0.33) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL14229219 0.85 MEN1 (0.35) MEN1KMT2ATP53HDAC8
SCHEMBL14229554 0.85 MEN1 (0.35) CYP1A2CYP2C19MEN1KMT2ATP53
SCHEMBL14229074 0.85 CYP1A2 (0.36) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL14201013 0.85 CYP1A2 (0.34) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL14229031 0.84 ALDH1A1 (0.44) MEN1KMT2AKDM4EALDH1A1TSHR
SCHEMBL14229068 0.83 CYP1A2 (0.35) CYP1A2CYP2D6CYP2C9CYP2C19NPSR1
SCHEMBL14228985 0.83 KMT2A (0.36) CYP1A2CYP2C9CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed