SCHEMBL14229304

SCHEMBL14229304

CCCC(=O)N(CCC)c1ccc(F)c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.49
NPSR1 Q6W5P4 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 3/20 0.38
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
LTB4R2 Q9NPC1 2/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 1/20 0.34
POLB P06746 2/20 0.34
APEX1 P27695 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MLYCD O95822 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229440 0.92 TP53 (0.47) TP53NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL14201015 0.85 NPSR1 (0.41) TP53NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL14229428 0.84 TP53 (0.50) TP53ALDH1A1LMNALTB4R2MEN1
SCHEMBL14229452 0.81 TP53 (0.50) TP53NPSR1ALDH1A1LMNAMEN1
SCHEMBL14229460 0.79 NPSR1 (0.37) TP53NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL14229074 0.78 CYP1A2 (0.36) TP53NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL14201035 0.78 MLYCD (0.38) TP53NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL14229265 0.77 CYP1A2 (0.39) TP53NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL14229264 0.77 TP53 (0.59) TP53ALDH1A1LMNALTB4R2MEN1
SCHEMBL14229061 0.76 TP53 (0.48) TP53ALDH1A1LMNALTB4R2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed