SCHEMBL14229504

SCHEMBL14229504

CCCCN(CCC)C(=O)OCCCl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.41
CA9 Q16790 3/20 0.41
CA1 P00915 2/20 0.41
MMP1 P03956 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP8 P22894 1/20 0.39
EGFR P00533 2/20 0.39
ERBB2 P04626 2/20 0.39
SIGMAR1 Q99720 2/20 0.36
ALDH1A1 P00352 2/20 0.35
CA2 P00918 1/20 0.35
DNM1 Q05193 1/20 0.34
TSHR P16473 2/20 0.33
ALDH2 P05091 1/20 0.33
MAPK1 P28482 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14228912 0.96 CA12 (0.44) CA12CA9CA1MMP1MMP2
SCHEMBL2478022 0.93 EGFR (0.42) CA12CA9CA1MMP1MMP2
SCHEMBL14229113 0.85 CA1 (0.36) CA12CA9CA1MMP1MMP2
SCHEMBL14200269 0.85 CA12 (0.36) CA12CA9CA1MMP1MMP2
SCHEMBL14230105 0.83 CA12 (0.37) CA12CA9CA1MMP1MMP2
SCHEMBL14229673 0.83 MMP1 (0.39) CA12CA9CA1MMP1MMP2
SCHEMBL8909554 0.83 ALDH1A1 (0.52) CA12CA9CA1ALDH1A1CA2
SCHEMBL19018673 0.83 CA12 (0.48) CA12CA9CA1MMP1MMP2
SCHEMBL65775 0.83 ALDH1A1 (0.52) CA12CA9CA1MMP1MMP2
SCHEMBL5158940 0.81 ALDH1A1 (0.47) CA12CA9CA1EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed