SCHEMBL14232129

SCHEMBL14232129

COBNCc1ccc(Cn2ccnc(N3CCN(CCOc4ccc(F)cc4)CC3)c2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.41
HTR1A P08908 7/20 0.41
HTR7 P34969 5/20 0.41
HTR6 P50406 4/20 0.41
DRD1 P21728 4/20 0.41
DRD3 P35462 4/20 0.41
HTR2A P28223 3/20 0.41
SIGMAR1 Q99720 1/20 0.39
MCHR1 Q99705 4/20 0.38
HRH3 Q9Y5N1 3/20 0.38
KCNH2 Q12809 1/20 0.38
DRD5 P21918 3/20 0.38
HRH1 P35367 2/20 0.38
ADRA2C P18825 1/20 0.38
HRH2 P25021 1/20 0.37
LTA4H P09960 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13633493 0.85 DRD2 (0.41) DRD2HTR1AHTR7HTR6DRD1
SCHEMBL13633485 0.84 DRD2 (0.47) DRD2HTR1AHTR7HTR6DRD1
SCHEMBL13633465 0.84 HTR1A (0.51) DRD2HTR1AHTR7DRD1DRD3
SCHEMBL13633487 0.82 DRD2 (0.43) DRD2HTR1AHTR7HTR6DRD1
SCHEMBL13633434 0.82 DRD2 (0.52) DRD2HTR1AHTR7DRD1DRD3
SCHEMBL13633492 0.77 DRD2 (0.45) DRD2HTR1AHTR7DRD1DRD3
SCHEMBL13633482 0.77 HTR1A (0.54) DRD2HTR1AHTR7DRD1DRD3
SCHEMBL13633481 0.77 DRD2 (0.48) DRD2HTR1AHTR7DRD1DRD3
SCHEMBL13633483 0.76 LTA4H (0.53) DRD2HTR1AHTR7DRD1DRD3
SCHEMBL2641162 0.70 HTR1A (0.43) DRD2HTR1AHTR7DRD1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007135131-A9 SUBSTITUTED PYRAZINONE DERIVATIVES FOR USE AS A MEDICINE JANSSEN PHARMACEUTICA NV (BE) 2008-04-03 WO disclosed