SCHEMBL142379

SCHEMBL142379

O=C(O)C1=NCCC1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835844 1.00
SCHEMBL4674692 0.92
SCHEMBL14398018 0.90 HPGD (0.42)
SCHEMBL3664692 0.81 TP53 (0.39)
SCHEMBL2546819 0.78 TP53 (0.30)
SCHEMBL329231 0.77
Hydrochloric Acid SCHEMBL14844794 0.75 NOS3 (0.48)
SCHEMBL31128189 0.73 ALDH1A1 (0.50)
SCHEMBL883443 0.72
SCHEMBL12762365 0.70 NOS3 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 71 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4181781-B1 BREATH-BASED THERAPEUTIC DRUG MONITORING METHOD UNIV KINDERSPITAL BEIDER BASEL (CH) 2026-05-20 EP disclosed
EP-4219735-B1 METHOD AND APPARATUS FOR ANALYTE DETECTION USING AN ELECTROCHEMICAL BIOSENSOR ABBOTT DIABETES CARE (US) 2026-04-01 EP disclosed
US-20250258146-A1 QUANTITATIVE DETECTION METHOD OF MULTIPLE METABOLITES IN BIOLOGICAL SAMPLE AND METABOLIC CHIP HUMAN METABOLOMICS INSTITUTE INC. (CN) 2025-08-14 US disclosed
CN-118005607-B Process for the preparation of (S) -nicotine from myosmine 扎诺普瑞玛生命科学有限公司 2025-06-17 CN disclosed
CN-113950534-B Method for producing L-type cyclic amino acid 株式会社API 2025-05-20 CN disclosed
EP-4538692-A2 METHOD AND APPARATUS FOR ANALYTE DETECTION USING AN ELECTROCHEMICAL BIOSENSOR Abbott Diabetes Care (US) 2025-04-16 EP disclosed
WO-2025072741-A1 PRESERVATIVES FOR MOLECULAR SAMPLE ANALYSIS WITH SAMPLE COLLECTION DEVICES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2025-04-03 WO disclosed
EP-4419487-A1 SYSTEMS AND METHODS FOR BIOREMEDIATION OF PER- AND POLYFLUOROALKYL SUBSTANCES AND 1,4-DIOXANE The Trustees Of Columbia University In The City Of New York (US) 2024-08-28 EP disclosed
CN-118005607-A Process for the preparation of (S) -nicotine from myosmine 扎诺普瑞玛生命科学有限公司 2024-05-10 CN disclosed
US-20230277125-A1 BREATH-BASED THERAPEUTIC DRUG MONITORING METHOD UNIVERSITÄTS-KINDERSPITAL BEIDER BASEL (CH) 2023-09-07 US disclosed
WO-2010048582-A1 BIOSYNTHETICALLY GENERATED PYRROLINE-CARBOXY-LYSINE AND SITE SPECIFIC PROTEIN MODIFICATIONS VIA CHEMICAL DERIVATIZATION OF PYRROLINE-CARBOXY-LYSINE AND PYRROLYSINE RESIDUES IRM LLC (BM) 2010-04-29 WO disclosed
WO-2010048582-A1 BIOSYNTHETICALLY GENERATED PYRROLINE-CARBOXY-LYSINE AND SITE SPECIFIC PROTEIN MODIFICATIONS VIA CHEMICAL DERIVATIZATION OF PYRROLINE-CARBOXY-LYSINE AND PYRROLYSINE RESIDUES IRM LLC (BM) 2010-04-29 WO disclosed
EP-2084519-A2 ADVANCED DRUG DEVELOPMENT AND MANUFACTURING Los Alamos National Security, LLC (US) 2009-08-05 EP disclosed
WO-2008127291-A2 ADVANCED DRUG DEVELOPMENT AND MANUFACTURING LOS ALAMOS NATIONAL SECURITY, LLC (US) 2008-10-23 WO disclosed
US-20080220441-A1 Advanced drug development and manufacturing THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2008-09-11 US disclosed
EP-1629092-A2 CRYSTALLOGRAPHIC STRUCTURE OF TRYPANOSOMA CRUZI PROLINE RACEMASE (TcPRACA) AND USES THEREOF INSTITUT PASTEUR (FR) 2006-03-01 EP disclosed
EP-1592788-A2 IDENTIFICATION AND CHARACTERIZATION OF RACEMASES, DEFINITION OF PROTEIN SIGNATURES, AND A TEST FOR DETECTING D-AMINO ACID AND FOR SCREENING MOLECULES CAPABLE OF INHIBITING THE ACTIVITY OF RACEMASE, ESPECIALLY PROLINE RACEMASE INSTITUT PASTEUR (FR) 2005-11-09 EP disclosed
WO-2004106506-A2 CRYSTALLOGRAPHIC STRUCTURE OF TRYPANOSOMA CRUZI PROLINE RACEMASE (TCPRACA) AND USES THEREOF INSTITUT PASTEUR (FR) 2004-12-09 WO disclosed
WO-2004072223-A2 IDENTIFICATION AND CHARACTERIZATION OF RACEMASES, DEFINITION OF PROTEIN SIGNATURES, AND A TEST FOR DETECTING D-AMINO ACID AND FOR SCREENING MOLECULES CAPABLE OF INHIBITING THE ACTIVITY OF RACEMASE, ESPECIALLY PROLINE RACEMASE INSTITUT PASTEUR (FR) 2004-08-26 WO disclosed
EP-0307390-A2 Chemical compound consisting of cis-3-hydroxyproline for therapeutic treatment, and process for its preparation MERCKLE GMBH (DE) 1989-03-15 EP disclosed