SCHEMBL14239052

SCHEMBL14239052

CC1(C)CCc2nc3cc(-c4cncc(F)c4)ccc3c(=O)n2C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.40
CYP11B1 P15538 1/20 0.40
RAB9A P51151 6/20 0.38
NPC1 O15118 5/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
DYRK1A Q13627 2/20 0.37
GSK3B P49841 1/20 0.37
LMNA P02545 1/20 0.37
PIK3CG P48736 1/20 0.36
ABL1 P00519 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
CTSD P07339 1/20 0.35
BACE1 P56817 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14239050 0.89 RAB9A (0.40) RAB9ANPC1SMN1; SMN2LMNACYP1A2
SCHEMBL6921870 0.88 RAB9A (0.40) RAB9ANPC1SMN1; SMN2LMNACYP1A2
SCHEMBL14239358 0.88 RAB9A (0.44) RAB9ANPC1SMN1; SMN2LMNACYP1A2
SCHEMBL14239051 0.85 RAB9A (0.40) RAB9ANPC1SMN1; SMN2LMNACYP1A2
SCHEMBL14238938 0.84 GRM2 (0.42) CYP11B2CYP11B1DYRK1AGSK3BCYP1A2
SCHEMBL14239808 0.84 RAB9A (0.41) RAB9ANPC1SMN1; SMN2LMNACYP1A2
SCHEMBL14239054 0.83 RAB9A (0.37) RAB9ANPC1SMN1; SMN2LMNACYP1A2
SCHEMBL15818303 0.83 GRM5 (0.46) RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL14239353 0.82 CYP3A4 (0.41) RAB9ANPC1SMN1; SMN2LMNACYP1A2
SCHEMBL14239132 0.82 ALDH1A1 (0.44) RAB9ANPC1SMN1; SMN2LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed