SCHEMBL14239115

SCHEMBL14239115

CCC1CCc2nc3cc(-c4ccccn4)cnc3c(=O)n2C1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 2/20 0.35
USP30 Q70CQ3 3/20 0.34
SMO Q99835 2/20 0.34
CYP3A4 P08684 1/20 0.33
TGFBR1 P36897 1/20 0.33
HCRTR1 O43613 5/20 0.33
HCRTR2 O43614 5/20 0.33
HTR6 P50406 1/20 0.32
PDE5A O76074 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA7 P36544 1/20 0.32
CHRNA4 P43681 1/20 0.32
CNR2 P34972 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14239108 0.91 SMO (0.39) METAP2USP30SMOCYP3A4TGFBR1
SCHEMBL14239107 0.87 USP30 (0.35) METAP2USP30CYP3A4TGFBR1CHRNB2
SCHEMBL14240248 0.84 SMO (0.36) METAP2USP30SMOCYP3A4TGFBR1
SCHEMBL14239116 0.83 NPC1 (0.36) METAP2TGFBR1HCRTR1HCRTR2CHRNB2
SCHEMBL6922373 0.82 MAPT (0.37) METAP2USP30TGFBR1CNR2HRH3
SCHEMBL15818511 0.81 POLB (0.36) HCRTR1
SCHEMBL6923220 0.81 MAPT (0.36) METAP2USP30CYP3A4TGFBR1CHRNB2
SCHEMBL14239112 0.80 METAP2 (0.35) METAP2USP30TGFBR1HCRTR1HCRTR2
SCHEMBL14239044 0.80 TGFBR1 (0.36) METAP2USP30TGFBR1HCRTR1HCRTR2
SCHEMBL14238857 0.79 METAP2 (0.34) METAP2USP30TGFBR1CHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed