SCHEMBL14239116

SCHEMBL14239116

CC1CCCc2nc3cc(-c4ccccn4)cnc3c(=O)n2C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
TDP1 Q9NUW8 2/20 0.36
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
LMNA P02545 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
TGFBR1 P36897 4/20 0.35
NSD2 O96028 1/20 0.35
CNR2 P34972 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
MAPT P10636 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14239107 0.94 USP30 (0.35) NPC1RAB9ATDP1ALDH1A1SMN1; SMN2
SCHEMBL6923220 0.88 MAPT (0.36) TGFBR1CNR2CHRNB2CHRNB4CHRNA3
SCHEMBL6920770 0.87 NPC1 (0.44) NPC1RAB9ATDP1ALDH1A1KDM4E
SCHEMBL6922373 0.85 MAPT (0.37) NPC1RAB9ATDP1ALDH1A1KDM4E
SCHEMBL14239109 0.84 CNR2 (0.37) NPC1RAB9ATDP1ALDH1A1KDM4E
SCHEMBL14239115 0.83 METAP2 (0.35) TGFBR1CNR2CHRNB2CHRNB4CHRNA3
SCHEMBL12059162 0.83 MEN1 (0.49) NPC1RAB9ATDP1ALDH1A1KDM4E
SCHEMBL6922971 0.82 MEN1 (0.51) NPC1RAB9ATDP1ALDH1A1KDM4E
SCHEMBL14239113 0.82 LMNA (0.39) LMNATGFBR1CNR2MAPTHRH3
SCHEMBL14238857 0.82 METAP2 (0.34) NPC1RAB9ATDP1TGFBR1NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed