SCHEMBL14239351

SCHEMBL14239351

CCC1(F)CCc2nc3cc(-c4ccccn4)cnc3c(=O)n2CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 2/20 0.35
NPC1 O15118 4/20 0.34
RAB9A P51151 4/20 0.34
TDP1 Q9NUW8 2/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
NSD2 O96028 1/20 0.33
TGFBR1 P36897 3/20 0.33
CNR2 P34972 2/20 0.33
ALDH1A1 P00352 3/20 0.32
TP53 P04637 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TNKS O95271 1/20 0.32
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
CNR1 P21554 1/20 0.32
KDM4E B2RXH2 3/20 0.32
ACHE P22303 2/20 0.32
USP2 O75604 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14238855 0.89 NPC1 (0.35) METAP2NPC1RAB9ATDP1HCRTR1
SCHEMBL14239311 0.88 NPC1 (0.36) METAP2NPC1RAB9ATDP1HCRTR1
SCHEMBL14239349 0.88 NPC1 (0.42) METAP2NPC1RAB9ATDP1NSD2
SCHEMBL6922660 0.82 AXL (0.35) METAP2NPC1RAB9ATDP1NSD2
SCHEMBL14239422 0.82 GRM5 (0.35) NPC1RAB9ATDP1HCRTR1NSD2
SCHEMBL14238857 0.81 METAP2 (0.34) METAP2NPC1RAB9ATDP1NSD2
SCHEMBL14238856 0.81 METAP2 (0.34) METAP2NPC1RAB9ATDP1HCRTR1
SCHEMBL12059162 0.81 MEN1 (0.49) NPC1RAB9ATDP1NSD2TGFBR1
SCHEMBL14239313 0.81 TGFBR1 (0.37) METAP2NPC1RAB9ATDP1HCRTR1
SCHEMBL14239315 0.80 TGFBR1 (0.35) METAP2NPC1RAB9ATDP1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed