SCHEMBL1427

SCHEMBL1427

CCCc1nc(C(F)(F)F)c(C=O)n1Cc1ccc(-c2ccccc2C(=O)O)cc1

nearest known ligand 0.76

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL671 0.86 PPARG (0.67) PPARG
SCHEMBL7359247 0.85 AGTR2 (0.67) PPARG
SCHEMBL306 0.81 AGTR1 (0.76)
SCHEMBL33 0.81 AGTR1 (0.75)
SCHEMBL9756284 0.80 AGTR1 (0.67) PPARG
SCHEMBL684085 0.80 AGTR1 (0.71) PPARG
SCHEMBL181 0.78 AGTR1 (0.73)
SCHEMBL29833187 0.77 PPARG (0.70) PPARG
SCHEMBL29833188 0.77 PPARG (0.70) PPARG
SCHEMBL8396958 0.77 PPARG (1.00) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019048-B1 USE OF AN ANGIOTENSIN II RECEPTOR ANTAGONIST FOR THE PREPARATION OF DRUGS TO INCREASE THE SURVIVAL RATE OF RENAL TRANSPLANT PATIENTS MERCK SHARP DOHME ITALIA S P A (IT) 2004-01-21 EP claimed
US-5155118-A Administering angiotensin inhibitor E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-10-13 US claimed
US-5153197-A Treatment of hypertension with angiotensin II blocking imidazoles E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-10-06 US claimed
US-5138069-A Treating hypertension and congestive heart failure E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-08-11 US claimed
US-5128355-A Hypotensive E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-07-07 US claimed
US-5663187-A ANTICHOLESTEROL AGENTS AND ENZYME INHIBITORS MERCK & CO., INC. (US) 1997-09-02 US disclosed