SCHEMBL1427142

SCHEMBL1427142

CSCc1cccc2c(C(c3ccc(Cl)cc3F)C(C)CCS(=O)(=O)O)c[nH]c12

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 3/20 0.34
GCGR P47871 2/20 0.33
NR3C2 P08235 1/20 0.32
ADRB3 P13945 6/20 0.31
CYP3A4 P08684 1/20 0.30
NOS1 P29475 1/20 0.30
CYP2C19 P33261 1/20 0.30
NOS2 P35228 1/20 0.30
ADRB1 P08588 3/20 0.30
ADRB2 P07550 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1349203 0.86 ADRB3 (0.34) GCGRADRB3ADRB1ADRB2
SCHEMBL1348878 0.84 NR3C1 (0.32) NR3C1NR3C2
SCHEMBL1348774 0.83 PNP (0.32)
SCHEMBL1350811 0.79 GPR84 (0.35)
SCHEMBL1349758 0.78 PNP (0.36) GCGRADRB3CYP3A4NOS1CYP2C19
SCHEMBL1427183 0.77 HDAC3 (0.36) NR3C1
SCHEMBL1349740 0.77 MEN1 (0.32) NR3C1NR3C2
SCHEMBL1426920 0.77 MGAM (0.37) NR3C1GCGR
SCHEMBL1349776 0.76 GPR84 (0.34)
SCHEMBL1349194 0.76 OPRM1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300423-A1 SUBSTITUTED 7-SULFANYLMETHYL, 7-SULFINYLMETHYL AND 7-SULFONYLMETHYL INDOLES AND USE THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2011-03-30 EP disclosed
WO-2009156072-A1 SUBSTITUTED 7-SULFANYLMETHYL, 7-SULFINYLMETHYL AND 7-SULFONYLMETHYL INDOLES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-12-30 WO disclosed