SCHEMBL14291379

SCHEMBL14291379

COc1cc2ccn(-c3ccc(N)cc3Cl)c2cc1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.40
MAPT P10636 5/20 0.39
KDM4E B2RXH2 3/20 0.39
RAD52 P43351 1/20 0.39
ALDH1A1 P00352 4/20 0.39
POLB P06746 1/20 0.39
HTT P42858 2/20 0.38
LMNA P02545 1/20 0.38
PRKCI P41743 1/20 0.37
GAA P10253 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP3A4 P08684 3/20 0.35
NFKB1 P19838 1/20 0.35
PMP22 Q01453 1/20 0.35
SUV39H2 Q9H5I1 1/20 0.35
TTBK1 Q5TCY1 1/20 0.35
TSHR P16473 2/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14291380 0.82 ROCK1 (0.51) MAPTKDM4ERAD52ALDH1A1POLB
SCHEMBL4578786 0.81 ROCK2 (0.45) POLBHTTCYP3A4TSHRMAPK1
SCHEMBL14291381 0.77 MAPT (0.42) NR4A1MAPTKDM4EALDH1A1POLB
SCHEMBL3749826 0.72 CYP3A4 (0.44) NR4A1MAPTKDM4ERAD52ALDH1A1
SCHEMBL29393582 0.68 MEN1 (0.57) NR4A1MAPTKDM4EALDH1A1HTT
SCHEMBL77110 0.68 MEN1 (0.57) NR4A1MAPTKDM4EALDH1A1HTT
SCHEMBL31554543 0.67 NCF1 (0.47) ROCK1
SCHEMBL22509234 0.66 PGK1 (0.48) PRKCIGAA
Hydrochloric Acid SCHEMBL6235400 0.66 MEN1 (0.55) NR4A1MAPTKDM4EALDH1A1HTT
SCHEMBL31116725 0.65 ROCK1 (0.47) MAPTKDM4EALDH1A1LMNACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008024978-A2 TETRAHYDROINDOLONE AND TETRAHYDROINDAZOLONE DERIVATIVES SERENEX, INC. (US) 2008-02-28 WO disclosed