SCHEMBL14293370

SCHEMBL14293370

Cn1nc(C=N)cc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.41
DDB1 Q16531 2/20 0.40
CRBN Q96SW2 2/20 0.40
RAB9A P51151 3/20 0.39
NPC1 O15118 2/20 0.39
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 4/20 0.38
HPGD P15428 3/20 0.38
HSD17B10 Q99714 1/20 0.38
KMT2A Q03164 2/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1780239 0.82 DDB1 (0.43) GRM5DDB1CRBNRAB9ANPC1
SCHEMBL21670888 0.77 NPC1 (0.57) RAB9ANPC1ALDH1A1HPGDKMT2A
SCHEMBL16386822 0.74 DDB1 (0.42) GRM5DDB1CRBNRAB9ANPC1
SCHEMBL680089 0.73 NPC1 (0.61) GRM5DDB1CRBNRAB9ANPC1
SCHEMBL822565 0.73 ALDH1A1 (0.53) DDB1CRBNALDH1A1KMT2AMAPT
SCHEMBL7371813 0.72 CYP1A2 (0.47) GRM5DDB1CRBNRAB9ANPC1
SCHEMBL20532607 0.72 KMT2A (0.44) GRM5DDB1CRBNRAB9ANPC1
SCHEMBL8525179 0.72 GRM5 (0.43) GRM5DDB1CRBNRAB9ANPC1
SCHEMBL3757964 0.72 DDB1 (0.43) GRM5DDB1CRBNRAB9ANPC1
SCHEMBL21670879 0.71 GRM5 (0.34) GRM5DDB1CRBNRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008019690-A1 SUBSTITUTED ACETYLENIC COMPOUNDS USEFUL FOR THE TREATMENT OF DISEASES LEO PHARMA A/S (DK) 2008-02-21 WO disclosed