SCHEMBL14301206

SCHEMBL14301206

COc1ccc(NS(=O)(=O)c2cccc3cccnc23)c(C(=O)O)c1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 7/20 0.67
KMT2A Q03164 7/20 0.67
ALDH1A1 P00352 3/20 0.67
MAPT P10636 1/20 0.67
HPGD P15428 1/20 0.67
NPSR1 Q6W5P4 1/20 0.67
TP53 P04637 1/20 0.64
HTT P42858 1/20 0.64
SLC40A1 Q9NP59 6/20 0.60
POLB P06746 1/20 0.59
TSHR P16473 1/20 0.58
MMP2 P08253 1/20 0.57
GLO1 Q04760 2/20 0.55
ATM Q13315 1/20 0.54
GAA P10253 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL498858 0.84 MMP2 (0.60) MEN1KMT2AALDH1A1SLC40A1POLB
SCHEMBL5597927 0.84 MEN1 (0.65) MEN1KMT2AALDH1A1SLC40A1POLB
SCHEMBL3982318 0.83 METAP2 (0.60) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL5072651 0.83 KCNA5 (0.78) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL5616231 0.83 KCNA5 (0.78) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL5072760 0.82 MEN1 (0.59) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL5074804 0.82 MEN1 (0.59) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL5072751 0.82 MEN1 (0.71) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL5072311 0.81 MEN1 (0.58) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL30854819 0.80 CXCR2 (0.77) MEN1KMT2AALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399423-B9 ANTHRANILIC ACID AMIDES WITH A HETEROARYLSULFONYL SIDE CHAIN, METHOD FOR THE PRODUCTION THEREOF, USE THEREOF AS A MEDICAMENT OR DIAGNOSTIC AGENT AND PHARMACEUTICAL PREPARATIONS CONTAINING SAID COMPOUNDS SANOFI AVENTIS DEUTSCHLAND (DE) 2008-02-27 EP disclosed
EP-1399423-B1 ANTHRANILIC ACID AMIDES WITH A HETEROARYLSULFONYL SIDE CHAIN, METHOD FOR THE PRODUCTION THEREOF, USE THEREOF AS A MEDICAMENT OR DIAGNOSTIC AGENT AND PHARMACEUTICAL PREPARATIONS CONTAINING SAID COMPOUNDS SANOFI AVENTIS DEUTSCHLAND (DE) 2007-11-14 EP disclosed
US-7235664-B2 Anthranilamides with heteroarylsulfonyl side chain, process of preparation, and use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-06-26 US disclosed
US-7235664-B2 Anthranilamides with heteroarylsulfonyl side chain, process of preparation, and use SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-06-26 US disclosed