SCHEMBL14304582

SCHEMBL14304582

COc1ccc2c(c1)c(I)cn2C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.47
HTR6 P50406 2/20 0.45
AKR1C2 P52895 2/20 0.43
PDE10A Q9Y233 1/20 0.41
MTNR1A P48039 6/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MTNR1B P49286 5/20 0.40
AKR1C4 P17516 1/20 0.39
PTGS1 P23219 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
RAB9A P51151 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NQO2 P16083 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29942639 1.00 AKR1C3 (0.47) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL29162329 0.90 HTR6 (0.40) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL18386657 0.85 AKR1C3 (0.48) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL29992656 0.84 AKR1C3 (0.47) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL1357445 0.84 AKR1C3 (0.47) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL29992688 0.84 AKR1C3 (0.47) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL14304584 0.83 AKR1C3 (0.61) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL29954772 0.83 AKR1C3 (0.46) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL1778702 0.83 AKR1C3 (0.46) AKR1C3HTR6AKR1C2PDE10AMTNR1A
SCHEMBL31555881 0.83 KDM4E (0.48) AKR1C3HTR6AKR1C2PDE10AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008014249-A2 IMPROVED PREPARATIONS OF 2 -SUBSTITUTED PYRROLO [2, 3-B] PYRAZINE ( 4, 7 -DIAZAINDOLE ) COMPOUNDS SANOFI-AVENTIS (FR) 2008-01-31 WO disclosed