SCHEMBL14307992

SCHEMBL14307992

NC(=O)c1cn(-c2ccccc2)nc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.54
PARP2 Q9UGN5 1/20 0.54
PARP3 Q9Y6F1 1/20 0.54
DGAT1 O75907 11/20 0.52
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.50
PKM P14618 1/20 0.50
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
GALR3 O60755 1/20 0.45
SCN9A Q15858 1/20 0.45
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 1/20 0.43
AURKA O14965 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL408273 0.88 DGAT1 (0.54) DGAT1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL4298033 0.85 DGAT1 (0.57) DGAT1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL17350704 0.85 DGAT1 (0.52) DGAT1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL4408386 0.85 SCN9A (0.46) PARP1PARP2PARP3DGAT1KDM4E
SCHEMBL10576877 0.81 MAPT (0.63) DGAT1KDM4EALDH1A1CA12CA1
SCHEMBL23212137 0.81 BCAT2 (0.45) PARP1DGAT1KDM4EALDH1A1CA12
SCHEMBL29370792 0.81 BCAT2 (0.45) PARP1DGAT1KDM4EALDH1A1CA12
SCHEMBL4484548 0.80 SCN9A (0.57) PARP1PARP2PARP3DGAT1SCN9A
SCHEMBL407255 0.79 DGAT1 (0.67) DGAT1
SCHEMBL16378282 0.79 DGAT1 (0.40) PARP1DGAT1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008011131-A2 AMIDE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-01-24 WO disclosed