SCHEMBL14309643

SCHEMBL14309643

O=c1c(Br)cc(CC2C=CC=CC2)cn1Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
MAPK10 P53779 2/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 2/20 0.36
THRB P10828 2/20 0.36
NPSR1 Q6W5P4 2/20 0.35
RECQL P46063 1/20 0.35
USP2 O75604 1/20 0.34
KDM4E B2RXH2 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
BRD4 O60885 3/20 0.34
TRIM24 O15164 1/20 0.34
BRD1 O95696 1/20 0.34
CCL2 P13500 1/20 0.34
TAF1 P21675 1/20 0.34
BRD2 P25440 1/20 0.34
SMARCA2 P51531 1/20 0.34
SMARCA4 P51532 1/20 0.34
BRPF1 P55201 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14308375 0.76 BRD4 (0.38) ALDH1A1MAPK10KDM4EBRD4TRIM24
SCHEMBL1191685 0.75 MAPK10 (0.45) ALDH1A1MAPK10MEN1KMT2AUSP2
SCHEMBL27704682 0.74 SIGMAR1 (0.48) SIGMAR1
SCHEMBL31621835 0.74 SIGMAR1 (0.48) SIGMAR1
SCHEMBL15816469 0.72 ADRA1D (0.51) ALDH1A1MAPK10MEN1KMT2AMAPT
SCHEMBL6235800 0.70 ADRA1D (0.48) ALDH1A1MAPK10MEN1KMT2AMAPT
SCHEMBL29001267 0.69 MAPK10 (0.51) ALDH1A1MAPK10MEN1KMT2AUSP2
SCHEMBL15815917 0.69 ALDH1A1 (0.55) ALDH1A1MEN1KMT2AMAPTNPSR1
Ethane SCHEMBL13370815 0.67 ALDH1A1 (0.51) ALDH1A1MAPK10MEN1KMT2AMAPT
SCHEMBL13689319 0.65 SIGMAR1 (0.39) ALDH1A1MAPTSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008010953-A2 PYRIDINONE DIKETO ACIDS: INHIBITORS OF HIV REPLICATION IN COMBINATION THERAPY UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2008-01-24 WO disclosed