SCHEMBL14310643

SCHEMBL14310643

COC(=O)c1nc2n(c(=O)c1O)CCCOC2(C)C

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.33
MAP3K12 Q12852 1/20 0.32
ALDH1A1 P00352 3/20 0.31
ERCC1 P07992 1/20 0.31
FEN1 P39748 1/20 0.31
ERCC4 Q92889 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1170436 0.93 NPSR1 (0.34) NPSR1MAP3K12ALDH1A1ERCC1FEN1
SCHEMBL12777960 0.87 KDM4E (0.36) ALDH1A1KDM4E
SCHEMBL1169614 0.86 MAP3K12 (0.34) MAP3K12ERCC1FEN1ERCC4
SCHEMBL1169812 0.80 L3MBTL1 (0.36) ALDH1A1KDM4EMAPK1
SCHEMBL14303989 0.79 KMT2A (0.36) NPSR1MAP3K12ALDH1A1KDM4EMAPK1
SCHEMBL14303988 0.79 HSD11B1 (0.35) NPSR1ALDH1A1ERCC1FEN1ERCC4
SCHEMBL5528388 0.78 ERCC1 (0.33) MAP3K12ERCC1FEN1ERCC4
SCHEMBL14511045 0.78 MAP3K12 (0.32) MAP3K12ERCC1FEN1ERCC4
SCHEMBL13917379 0.76 KCNH2 (0.54) NPSR1ALDH1A1ERCC1FEN1ERCC4
SCHEMBL13917632 0.74 KCNK3 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008002959-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-01-03 WO disclosed