Mosapride

Mosapride

SCHEMBL14320968

CCOc1cc(N)c(Cl)cc1C(=O)NCC1CN(Cc2ccc(F)cc2)CCO1.O.O=C(O)CC(O)(CC(=O)O)C(=O)O

nearest known ligand 0.84

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HTR3AHTR3BHTR3CHTR3DHTR3EHTR4

The experimentally established mechanism targets of Mosapride. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 known ✓ Q13639 2/20 0.51
DRD3 P35462 4/20 0.84
MEN1 O00255 1/20 0.84
LMNA P02545 1/20 0.84
CYP1A2 P05177 1/20 0.84
CYP3A4 P08684 1/20 0.84
HTR1A P08908 1/20 0.84
ADRA2A P08913 1/20 0.84
ADORA3 P0DMS8 1/20 0.84
CYP2C9 P11712 1/20 0.84
ADRA2B P18089 1/20 0.84
HTR2C P28335 1/20 0.84
SLC6A4 P31645 1/20 0.84
CYP2C19 P33261 1/20 0.84
HTR2B P41595 1/20 0.84
KMT2A Q03164 1/20 0.84
KCNH2 Q12809 1/20 0.84
SIGMAR1 Q99720 1/20 0.84
DRD4 P21917 12/20 0.46
DRD2 P14416 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mosapride SCHEMBL6227414 1.00 DRD3 (0.84) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL30450705 1.00 DRD3 (0.84) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL1098769 1.00 DRD3 (0.84) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL8462520 0.99 DRD3 (0.85) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL258620 0.99 DRD3 (0.85) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL2369236 0.92 DRD3 (0.98) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL6229365 0.92 DRD3 (0.91) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL29400580 0.91 DRD3 (1.00) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL6228981 0.91 DRD3 (1.00) DRD3MEN1LMNACYP1A2CYP3A4
Mosapride SCHEMBL16417 0.91 DRD3 (1.00) DRD3MEN1LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12582606-B2 Tablet and method for producing tablet SUNSHO PHARMACEUTICAL CO., LTD. (JP) 2026-03-24 US disclosed
WO-2025047788-A1 FILM PREPARATION HAVING ADHESIVENESS TO INSIDE OF ANIMAL ORAL CAVITY 株式会社ペティーナ 2025-03-06 WO disclosed
WO-2025047787-A1 FILM PREPARATION CAPABLE OF ADHERING TO ANIMAL ORAL CAVITIES 株式会社ペティーナ 2025-03-06 WO disclosed
US-20240016745-A1 TIMED-ELUTION MASKING PARTICLES AND ORAL PHARMACEUTICAL COMPOSITION CONTAINING THE SAME TOWA PHARMACEUTICAL CO., LTD. (JP) 2024-01-18 US disclosed
EP-4260847-A1 TIMED-ELUTION MASKING PARTICLES AND ORAL PHARMACEUTICAL COMPOSITION CONTAINING SAME TOWA PHARMACEUTICAL CO., LTD. (JP) 2023-10-18 EP disclosed
US-20220218616-A1 TABLET AND METHOD FOR PRODUCING TABLET SUNSHO PHARMACEUTICAL CO., LTD. (JP) 2022-07-14 US disclosed
US-11000481-B2 Composite preparation of mosapride and rabeprazole KOREA UNITED PHARM. INC. (KR) 2021-05-11 US disclosed
US-10746721-B2 Method for rapid testing allergy Shibaguchi, Hirotomo (JP) 2020-08-18 US disclosed
US-10746722-B2 Method for rapid testing allergy Shibaguchi, Hirotomo (JP) 2020-08-18 US disclosed
US-20190265225-A1 METHOD FOR RAPID TESTING ALLERGY SHIBAGUCHI HIROTOMO (JP) 2019-08-29 US disclosed
US-20190265224-A1 METHOD FOR RAPID TESTING ALLERGY SHIBAGUCHI HIROTOMO (US) 2019-08-29 US disclosed
US-10324079-B2 Method for rapid testing allergy Shibaguchi, Hirotomo (JP) 2019-06-18 US disclosed
CN-108289849-A Compound preparation of mosapride and rabeprazole 韩国联合制药株式会社 2018-07-17 CN disclosed
US-20180177731-A1 Composite Preparation of Mosapride and Rabeprazole KOREA UNITED PHARM. INC. (KR) 2018-06-28 US disclosed
EP-2975403-B1 RAPID ALLERGY TESTING METHOD SHIBAGUCHI HIROTOMO (JP) 2018-05-02 EP disclosed
US-20160069858-A1 RAPID ALLERGY TESTING METHOD Shibaguchi, Hirotomo (JP) 2016-03-10 US disclosed
EP-2975403-A1 RAPID ALLERGY TESTING METHOD Shibaguchi, Hirotomo (JP) 2016-01-20 EP disclosed
EP-2543366-A1 FILM PREPARATION CONTAINING MEDICAMENT WITH UNPLEASANT TASTE Kyukyu Pharmaceutical Co., Ltd. (JP) 2013-01-09 EP disclosed
US-20120328675-A1 FILM PREPARATION CONTAINING MEDICAMENT WITH UNPLEASANT TASTE KOWA CO., LTD. (JP) 2012-12-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12582606-B2 Tablet and method for producing tablet GRHPR, RCC1, KIT HTR4 1846/4885DRD3 4564/4885MEN1 3180/4885
US-20180177731-A1 Composite Preparation of Mosapride and Rabeprazole MLNR, RAB14, RAB29 HTR4 180/4885DRD3 1874/4885MEN1 1805/4885
US-11000481-B2 Composite preparation of mosapride and rabeprazole MLNR, RAB14, RAB29 HTR4 180/4885DRD3 1874/4885MEN1 1805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.