SCHEMBL14347495

SCHEMBL14347495

COc1cccc2c(C(C)(C)C)nc(=O)oc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 9/20 0.49
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 3/20 0.49
LMNA P02545 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
CYP2A6 P11509 1/20 0.45
HPGD P15428 2/20 0.45
MAPT P10636 2/20 0.45
CYP3A4 P08684 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
TNKS O95271 1/20 0.41
PARP1 P09874 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14347463 0.84 PRKDC (0.39) MAOAALDH1A1KDM4ELMNANPC1
SCHEMBL14347531 0.81 MAOA (0.33) MAOAALDH1A1KDM4ELMNANPC1
SCHEMBL14347475 0.79 HTR1B (0.49) ALDH1A1KDM4ELMNAMAPTKMT2A
SCHEMBL14347543 0.79 TNKS (0.39) ALDH1A1NPC1RAB9AMAPTCA12
SCHEMBL14347431 0.78 NPC1 (0.39) ALDH1A1KDM4ELMNANPC1RAB9A
SCHEMBL14347527 0.77 LOXL2 (0.43) PRKDC
SCHEMBL14374844 0.77 MAOA (0.49) MAOAALDH1A1KDM4ELMNANPC1
SCHEMBL14347415 0.77 ELANE (0.35) ALDH1A1KDM4ERAB9ACA1CA2
SCHEMBL14347532 0.76 CYP1A2 (0.50) ALDH1A1KDM4EMAPTHSD17B10MEN1
SCHEMBL14347473 0.75 PRKDC (0.59) KDM4EPRKDCSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7312211-B2 Pryanone compounds useful as reversible inhibitors of cysteine proteases BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2007-12-25 US disclosed