SCHEMBL14347463

SCHEMBL14347463

COCCOc1cccc2c(C(C)(C)C)nc(=O)oc12

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.39
KDM1A O60341 1/20 0.37
CNR2 P34972 2/20 0.36
MAOA P21397 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.34
F2RL3 Q96RI0 2/20 0.34
SIGMAR1 Q99720 1/20 0.33
CYP2A6 P11509 1/20 0.33
KCNA5 P22460 1/20 0.33
CSF1R P07333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14347475 0.85 HTR1B (0.49) PRKDCKDM4EALDH1A1LMNACSF1R
SCHEMBL14347495 0.84 MAOA (0.49) PRKDCMAOAKDM4ENPC1ALDH1A1
SCHEMBL14347527 0.82 LOXL2 (0.43) PRKDCLOXL2
SCHEMBL14347532 0.82 CYP1A2 (0.50) PRKDCKDM4EALDH1A1
SCHEMBL14374658 0.81 PRKDC (0.39) PRKDCKDM1ACNR2MAOAKDM4E
SCHEMBL14347473 0.81 PRKDC (0.59) PRKDCCNR2KDM4ESIGMAR1
SCHEMBL14347474 0.80 PRKDC (0.48) PRKDCSIGMAR1
SCHEMBL14347531 0.75 MAOA (0.33) PRKDCMAOAKDM4ENPC1ALDH1A1
SCHEMBL14347543 0.73 TNKS (0.39) NPC1ALDH1A1RAB9A
SCHEMBL14347461 0.72 APP (0.45) KDM4ENPC1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7312211-B2 Pryanone compounds useful as reversible inhibitors of cysteine proteases BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2007-12-25 US disclosed