SCHEMBL14360997

SCHEMBL14360997

Cc1cc[nH]c1C(=O)Nc1ccc(-c2sc(-c3ccno3)cc2C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.40
GRM1 Q13255 1/20 0.37
KMT2A Q03164 6/20 0.35
MEN1 O00255 5/20 0.35
ATM Q13315 1/20 0.35
GAA P10253 1/20 0.35
GFER P55789 1/20 0.35
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPT P10636 5/20 0.34
LRRK2 Q5S007 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
RXFP1 Q9HBX9 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KCNJ1 P48048 2/20 0.34
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8233130 0.82 ALOX15 (0.46) POLBKMT2AMEN1ATMGAA
SCHEMBL2891375 0.81 IL2 (0.46) POLBKMT2AMEN1LMNASMN1; SMN2
SCHEMBL14360818 0.80 POLB (0.51) POLBKMT2AMEN1GAAHPGD
SCHEMBL5030789 0.80 POLB (0.40) POLBKMT2AMEN1ATMGAA
SCHEMBL5033820 0.79 LMNA (0.49) POLBKMT2AMEN1ATMHPGD
SCHEMBL14360834 0.79 POLB (0.39) POLBKMT2AMEN1ATMGAA
SCHEMBL5030892 0.79 POLB (0.39) POLBKMT2AMEN1ATMGAA
SCHEMBL14360910 0.78 LRRK2 (0.42) POLBKMT2AMEN1ATMGAA
SCHEMBL14361068 0.78 POLB (0.47) POLBGRM1KMT2AMEN1HPGD
SCHEMBL2889603 0.76 KMT2A (0.43) POLBKMT2AMEN1MAPTESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070275960-A1 Phenyl and pyridyl compounds for inflammation and immune-related uses SYNTA PHARMACEUTICALS CORP. (US) 2007-11-29 US disclosed
US-20070275960-A1 Phenyl and pyridyl compounds for inflammation and immune-related uses SYNTA PHARMACEUTICALS CORP. (US) 2007-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275960-A1 Phenyl and pyridyl compounds for inflammation and immune-related uses NLRP3, CCR1, NLRP1 POLB 4194/4885GRM1 3684/4885KMT2A 3327/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.