SCHEMBL14363333

SCHEMBL14363333

Cc1ccc(O)c(C(=O)Nc2cc(O)c(O)c(O)c2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 6/20 0.67
TMPRSS4 Q9NRS4 4/20 0.67
PLAU P00749 2/20 0.63
F2 P00734 1/20 0.61
F10 P00742 1/20 0.61
PLAT P00750 1/20 0.61
GRM5 P41594 1/20 0.55
CSNK2A1 P68400 1/20 0.53
RAB9A P51151 3/20 0.53
NPC1 O15118 2/20 0.53
LMNA P02545 2/20 0.53
HSD17B10 Q99714 2/20 0.53
TP53 P04637 1/20 0.53
NFKB1 P19838 1/20 0.53
HTT P42858 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
P2RX4 Q99571 2/20 0.51
P2RX7 Q99572 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14363179 0.87 PLAU (0.65) P2RX1TMPRSS4PLAUF2F10
SCHEMBL21021862 0.86 PLAU (0.73) P2RX1TMPRSS4PLAUF2F10
SCHEMBL330475 0.84 P2RX1 (0.74) P2RX1TMPRSS4PLAUF2F10
SCHEMBL23336137 0.84 TMPRSS4 (0.63) P2RX1TMPRSS4PLAUF2F10
SCHEMBL6285639 0.83 TMPRSS4 (0.67) P2RX1TMPRSS4PLAUF2F10
SCHEMBL14363184 0.83 PLAU (0.69) P2RX1TMPRSS4PLAUF2F10
SCHEMBL14363264 0.81 KMT2A (0.60) P2RX1TMPRSS4PLAUF2F10
SCHEMBL330257 0.81 P2RX1 (0.77) P2RX1TMPRSS4PLAUF2F10
SCHEMBL19040075 0.81 PLAU (0.66) P2RX1TMPRSS4PLAUF2F10
SCHEMBL24460276 0.81 P2RX1 (0.77) P2RX1TMPRSS4PLAUF2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070276011-A1 Plasminogen Activator Inhibitor-1 Inhibitor INSTITUTE OF MEDICINAL MOLECULAR DESIGN. INC. (JP) 2007-11-29 US disclosed
US-20070276011-A1 Plasminogen Activator Inhibitor-1 Inhibitor INSTITUTE OF MEDICINAL MOLECULAR DESIGN. INC. (JP) 2007-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070276011-A1 Plasminogen Activator Inhibitor-1 Inhibitor SERPINE1, SERPINC1, SERPINB1 P2RX1 4478/4885TMPRSS4 342/4885PLAU 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.