SCHEMBL14366283

SCHEMBL14366283

O=C(Cc1ccc(F)cc1)NC(=O)Nc1ccc(Oc2ccnc(NC(=O)NCCCN3CCOCC3)c2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.47
EPHX2 P34913 4/20 0.46
CSF1R P07333 3/20 0.46
MET P08581 3/20 0.46
PDGFRB P09619 3/20 0.46
PDGFRA P16234 3/20 0.46
FLT3 P36888 3/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TACR2 P21452 2/20 0.44
TP53 P04637 1/20 0.44
FLT1 P17948 2/20 0.44
FLT4 P35916 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
RAF1 P04049 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14366284 0.92 MET (0.48) KDRCSF1RMETPDGFRBPDGFRA
SCHEMBL4323368 0.88 KDR (0.51) KDREPHX2METLMNAKMT2A
SCHEMBL4329648 0.87 L3MBTL1 (0.49) EPHX2LMNAKMT2ASMN1; SMN2TACR2
SCHEMBL14366285 0.82 KDR (0.45) KDRCSF1RMETPDGFRBPDGFRA
SCHEMBL14391787 0.82 MET (0.47) KDRCSF1RMETPDGFRBPDGFRA
SCHEMBL4333183 0.81 CA12 (0.48) KDREPHX2LMNAKMT2ASMN1; SMN2
SCHEMBL14366282 0.81 MET (0.46) KDRCSF1RMETPDGFRBPDGFRA
SCHEMBL4330370 0.80 MAPT (0.48) KDRMETPDGFRBFLT3LMNA
SCHEMBL4326460 0.79 KDR (0.42) KDRMETKMT2AFLT1FLT4
SCHEMBL4329670 0.79 L3MBTL1 (0.47) KDRLMNAKMT2ASMN1; SMN2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070270421-A1 Novel pyridine Derivative and Pyrimidine Derivative (1) EISAI R&D MANAGEMENT CO., LTD. (JP) 2007-11-22 US disclosed
US-20070270421-A1 Novel pyridine Derivative and Pyrimidine Derivative (1) EISAI R&D MANAGEMENT CO., LTD. (JP) 2007-11-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070270421-A1 Novel pyridine Derivative and Pyrimidine Derivative (1) HGF, MET, FLT1 KDR 7/4885EPHX2 2388/4885CSF1R 29/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.