SCHEMBL14367172

SCHEMBL14367172

POC/C=C/CN1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 7/20 0.63
LMNA P02545 5/20 0.63
HIF1A Q16665 4/20 0.63
OPRM1 P35372 4/20 0.63
CYP3A4 P08684 3/20 0.63
CYP2D6 P10635 3/20 0.63
NPSR1 Q6W5P4 3/20 0.63
MAPK1 P28482 3/20 0.63
CYP1A2 P05177 2/20 0.63
CYP2C9 P11712 2/20 0.63
CHRM2 P08172 2/20 0.63
CHRM4 P08173 2/20 0.63
HTR1A P08908 2/20 0.63
CHRM5 P08912 2/20 0.63
ADRA2A P08913 2/20 0.63
ADORA3 P0DMS8 2/20 0.63
CHRM1 P11229 2/20 0.63
DRD2 P14416 2/20 0.63
ADRA2B P18089 2/20 0.63
ADRA2C P18825 2/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1137893 0.81 OPRD1 (0.68) OPRD1LMNAHIF1AOPRM1CYP3A4
SCHEMBL9837345 0.81 OPRD1 (0.68) OPRD1LMNAHIF1AOPRM1CYP3A4
SCHEMBL1137896 0.81 OPRD1 (0.68) OPRD1LMNAHIF1AOPRM1CYP3A4
SCHEMBL9837343 0.81 OPRD1 (0.68) OPRD1LMNAHIF1AOPRM1CYP3A4
SCHEMBL1138084 0.80 NPC1 (0.60) OPRD1LMNAHIF1AOPRM1CYP3A4
SCHEMBL1138082 0.80 NPC1 (0.60) OPRD1LMNAHIF1AOPRM1CYP3A4
SCHEMBL6554369 0.80 OPRD1 (0.56) OPRD1LMNAHIF1AOPRM1CYP3A4
Hydrochloric Acid SCHEMBL1138342 0.79 HRH1 (0.58) OPRD1LMNAHIF1AOPRM1CYP3A4
Hydrochloric Acid SCHEMBL1138343 0.79 HRH1 (0.58) OPRD1LMNAHIF1AOPRM1CYP3A4
SCHEMBL14367175 0.78 OPRD1 (0.54) OPRD1LMNAHIF1AOPRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7297697-B2 with alkenyl moiety substituted at the 1-position of the piperazine unit; useful in the treatment of histamine mediated diseases SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2007-11-20 US disclosed