SCHEMBL14367752

SCHEMBL14367752

Cc1cccc(O)c1-c1nc2c(-c3nc4c(C(=O)O)cccc4o3)cccc2o1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 3/20 0.60
MYC P01106 1/20 0.46
IDO1 P14902 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
AGPAT2 O15120 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
TYMS P04818 1/20 0.37
IKBKB O14920 1/20 0.36
G6PD P11413 1/20 0.36
CASP7 P55210 1/20 0.36
CASP6 P55212 1/20 0.36
HTR3A P46098 2/20 0.36
KCNH2 Q12809 2/20 0.36
MCL1 Q07820 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29885350 1.00 TOP2A (0.60) TOP2AMYCIDO1MAOAMAOB
SCHEMBL2955256 0.86 MYC (0.49) TOP2AMYCIDO1MAOAMAOB
SCHEMBL14367754 0.85 TOP2A (0.75) TOP2AIDO1MAOAMAOBKDM4E
SCHEMBL3401507 0.83 TOP2A (0.58) TOP2AMYCIDO1MAOAMAOB
SCHEMBL2959863 0.82 TOP2A (0.70) TOP2AIDO1MAOAMAOBKDM4E
SCHEMBL10731139 0.78 TOP2A (0.55) TOP2AMYCAGPAT2KDM4EALDH1A1
SCHEMBL12807868 0.77 TOP2A (0.72) TOP2AAGPAT2KDM4EALDH1A1HSD17B10
SCHEMBL11979724 0.75 TOP2A (1.00) TOP2AAGPAT2KDM4EALDH1A1HPGD
SCHEMBL29354263 0.75 TOP2A (1.00) TOP2AAGPAT2KDM4EALDH1A1HPGD
SCHEMBL17929359 0.75 TOP2A (0.78) TOP2AAGPAT2KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294643-B2 UK-1 analogues: methods of preparation and use BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2007-11-13 US disclosed
US-7294643-B2 UK-1 analogues: methods of preparation and use BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2007-11-13 US disclosed