SCHEMBL1438281

SCHEMBL1438281

COc1ccc(Cl)cc1-c1cnn(-c2ccccc2)c1-c1cccc(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.54
RAB9A P51151 4/20 0.54
ALDH1A1 P00352 4/20 0.51
MAPT P10636 4/20 0.51
GAA P10253 4/20 0.51
HPGDS O60760 1/20 0.51
ATM Q13315 2/20 0.48
FYN P06241 1/20 0.46
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
MCL1 Q07820 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PDE4B Q07343 2/20 0.41
HPGD P15428 3/20 0.41
KDM4E B2RXH2 2/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1436956 0.90 PIP4K2A (0.44) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL10002437 0.76 MDM2 (0.48) ALDH1A1MAPTKMT2ANPSR1HPGD
SCHEMBL9893767 0.76 MDM2 (0.47) ALDH1A1MAPTKMT2ANPSR1HPGD
Lithium SCHEMBL9893769 0.76 MDM2 (0.47) ALDH1A1MAPTKMT2ANPSR1HPGD
Lithium Ion SCHEMBL9893768 0.74 TUBB4A (0.41) ALDH1A1MAPTKMT2ANPSR1TUBB4A
SCHEMBL5099550 0.73 PDE4D (0.56) NPC1ALDH1A1MAPTFYNPDE4B
SCHEMBL8765024 0.72 RAB9A (0.69) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL3759371 0.72 PTGDR2 (0.57) ALDH1A1KMT2AMEN1NPSR1HPGD
SCHEMBL29634149 0.72 PTGDR2 (0.57) ALDH1A1KMT2AMEN1NPSR1HPGD
SCHEMBL28301005 0.71 NPC1 (0.47) NPC1RAB9AALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011023677-A1 TETRA-SUBSTITUTED HETEROARYL COMPOUNDS AND THEIR USE AS MDM2 AND/OR MDM4 MODULATORS NOVARTIS AG (CH) 2011-03-03 WO disclosed