SCHEMBL14397487

SCHEMBL14397487

O=Cc1occc1-c1ccoc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 3/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
ESR1 P03372 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
APEX1 P27695 1/20 0.34
MAPK1 P28482 1/20 0.34
ESR2 Q92731 1/20 0.34
ACLY P53396 1/20 0.32
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
HSD17B10 Q99714 1/20 0.31
AGTR1 P30556 1/20 0.30
AGTR2 P50052 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14398057 0.77 POLB (0.50) KMT2AL3MBTL1POLBMAPK1ALDH1A1
SCHEMBL14397414 0.75 KMT2A (0.34) KMT2ATDP1L3MBTL1ESR1TP53
SCHEMBL14397443 0.75 POLB (0.34) KMT2ATDP1L3MBTL1TP53POLB
SCHEMBL14398161 0.75 PRKDC (0.33) KMT2ATDP1L3MBTL1ESR1TP53
SCHEMBL14397491 0.75 GPR35 (0.35) KMT2AL3MBTL1ALDH1A1
SCHEMBL14397520 0.75 CYP2C9 (0.34) POLBKDM4E
SCHEMBL8441952 0.74 KEAP1 (0.38) KMT2ATDP1L3MBTL1POLBALDH1A1
SCHEMBL11403524 0.73 APP (0.36) MAPK1ALDH1A1KDM4E
SCHEMBL14398163 0.73 KEAP1 (0.39) KMT2APOLBALDH1A1KDM4EHSD17B10
SCHEMBL14397519 0.73 CSNK2A1 (0.44) KMT2AL3MBTL1TP53POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007117180-A1 AZAHETEROCYCLES, COMBINATORY LIBRARY, FOCUSED LIBRARY, PHARMACEUTICAL COMPOSITION AND METHODS FOR THE PRODUCTION THEREOF 'CHEMICAL DIVERSITY RESEARCH INSTITUTE' LTD. (RU) 2007-10-18 WO disclosed