SCHEMBL14409100

SCHEMBL14409100

Cc1nnc(Sc2ccnc3ccccc23)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
MAPK1 P28482 1/20 0.49
PAX8 Q06710 1/20 0.49
ATM Q13315 1/20 0.49
MAPT P10636 4/20 0.42
GFER P55789 1/20 0.42
UBE2N P61088 1/20 0.42
POLB P06746 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 3/20 0.40
HPGD P15428 4/20 0.39
KDM4E B2RXH2 3/20 0.39
LMNA P02545 3/20 0.39
ABL1 P00519 1/20 0.39
RIN1 Q13671 1/20 0.39
USP2 O75604 1/20 0.39
ALOX15 P16050 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1821527 0.82 NPSR1 (0.63) PKMNPSR1MAPK1PAX8ATM
SCHEMBL1821065 0.82 MAPK1 (0.43) PKMNPSR1MAPK1PAX8ATM
SCHEMBL13791595 0.79 NPSR1 (0.75) PKMNPSR1MAPK1PAX8ATM
SCHEMBL13065100 0.75 LOXL2 (0.40) PKMNPSR1MAPK1PAX8ATM
SCHEMBL12656711 0.72 SMN1; SMN2 (0.60) PKMNPSR1MAPK1ATMMAPT
SCHEMBL12656928 0.72 HTT (0.44) MAPK1PAX8MAPTPOLBNPC1
SCHEMBL14409077 0.72 KMT2A (0.57) MAPK1NPC1RAB9AALDH1A1HPGD
SCHEMBL12657084 0.72 GLS (0.44) MAPK1MAPTPOLBNPC1RAB9A
SCHEMBL12656688 0.72 SMN1; SMN2 (0.56) NPSR1NPC1RAB9AALDH1A1HPGD
SCHEMBL12656927 0.71 RAB9A (0.41) PKMNPSR1MAPK1PAX8ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7271179-B2 Inhibitors of JAK protein kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-09-18 US disclosed