SCHEMBL14412293

SCHEMBL14412293

O=C(NCCN1CCCC1)c1ccc(-c2cc(C(F)(F)F)n(CF)n2)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
ALDH1A1 P00352 4/20 0.43
EPHX2 P34913 3/20 0.41
HDAC3 O15379 2/20 0.41
HDAC4 P56524 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC7 Q8WUI4 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC9 Q9UKV0 2/20 0.41
HDAC5 Q9UQL6 2/20 0.41
NCOR2 Q9Y618 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1594477 0.88 ALDH1A1 (0.57) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL1593887 0.87 ALDH1A1 (0.56) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL9966087 0.84 KMT2A (0.46) ALDH1A1MEN1KMT2AHTTL3MBTL1
SCHEMBL1593693 0.82 ALDH1A1 (0.55) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL1593840 0.80 ALDH1A1 (0.54) ALDH1A1EPHX2MEN1KMT2AHTT
SCHEMBL9966059 0.79 NPC1 (0.48) ALDH1A1CYP1A2CYP2D6CYP2C9MEN1
SCHEMBL14412372 0.78 ALDH1A1 (0.42) ALDH1A1HDAC3HDAC4HDAC1HDAC7
SCHEMBL9966063 0.77 KMT2A (0.53) ALDH1A1CYP1A2CYP2C9MEN1KMT2A
SCHEMBL9966057 0.77 KMT2A (0.53) ALDH1A1CYP1A2CYP2C9MEN1KMT2A
SCHEMBL14960353 0.76 ALDH1A1 (0.44) ALDH1A1HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007100851-A1 THERAPEUTIC COMPOUNDS HELICON THERAPEUTICS, INC. (US) 2007-09-07 WO disclosed