SCHEMBL14415552

SCHEMBL14415552

CCCOC1(c2ccc(Cl)c(Cl)c2)CCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.46
OPRM1 P35372 1/20 0.40
TACR1 P25103 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
GPR183 P32249 1/20 0.38
USP30 Q70CQ3 1/20 0.37
RORC P51449 1/20 0.37
SCD5 Q86SK9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13544004 0.94 CCR5 (0.46) CCR5OPRM1TACR1
SCHEMBL5510972 0.88 CCR5 (0.44) CCR5OPRM1TACR1PDE4APDE4B
SCHEMBL4680501 0.86 CCR5 (0.45) CCR5OPRM1TACR1PDE4APDE4B
SCHEMBL13543990 0.81 CCR5 (0.44) CCR5TACR1
SCHEMBL27228860 0.79 OPRM1 (0.46) CCR5OPRM1TACR1USP30RORC
SCHEMBL13543991 0.79 CCR5 (0.43) CCR5TACR1
SCHEMBL8563070 0.79 CCR5 (0.41) CCR5PDE4APDE4BPDE4CPDE4D
SCHEMBL3118407 0.79 CCR5 (0.47) CCR5TACR1USP30RORCSCD5
SCHEMBL1280507 0.79 USP2 (0.41) CCR5OPRM1
SCHEMBL14415546 0.79 CCR5 (0.51) CCR5OPRM1TACR1PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7271172-B2 Pyrrolidine and azetidine compounds as CCR5 antagonists SMITHKLINE BEECHAM CORPORATION (US) 2007-09-18 US disclosed