SCHEMBL144309

SCHEMBL144309

Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 1.00
ALDH1A1 P00352 2/20 1.00
GAA P10253 2/20 1.00
HPGD P15428 2/20 1.00
CASP1 P29466 2/20 1.00
CASP7 P55210 2/20 1.00
HSD17B10 Q99714 2/20 1.00
MEN1 O00255 1/20 1.00
SRC P12931 1/20 1.00
KMT2A Q03164 1/20 1.00
ATM Q13315 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
TLR9 Q9NR96 1/20 1.00
HSD17B3 P37058 1/20 0.67
AR P10275 12/20 0.58
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
GLA P06280 1/20 0.58
CA9 Q16790 1/20 0.58
MCL1 Q07820 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29356441 1.00 KDM4E (1.00) KDM4EALDH1A1GAAHPGDCASP1
Glycine SCHEMBL9259892 0.89 KDM4E (0.79) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL1771156 0.87 KDM4E (0.77) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL7973305 0.87 KDM4E (0.77) KDM4EALDH1A1GAAHPGDCASP1
Alanine SCHEMBL15556780 0.87 KDM4E (0.75) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL29156864 0.83 KDM4E (0.71) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL4620259 0.82 KDM4E (0.68) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL15842662 0.81 HSD17B3 (0.69) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL12611304 0.80 ALDH1A1 (0.67) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL307508 0.80 HSD17B3 (1.00) KDM4EALDH1A1GAAHPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3150 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12630857-B2 Biological indicator for determining the efficacy of a steam or heat sterilization process and its method of use TERRAGENE LLC (US) 2026-05-19 US claimed
EP-4731992-A1 GREEN ENERGY SOURCES AUTHENTICATION AND COMPLIANCE TESTING Authentix, Inc. (US) 2026-04-29 EP claimed
EP-4677362-A1 ENZYME LINKED IMMUNOASSAY WITH DIFFUSION RATE LIMITING MEDIUM Elleon Biotech Limited (HK) 2026-01-14 EP claimed
WO-2025234889-A1 METHOD FOR MANUFACTURING CARBON QUANTUM DOTS WITH A SHIFTED FLUORESCENCE EMISSION SPECTRUM Politechnika Krakowska im.Tadeusza Kościuszki (PL) 2025-11-13 WO claimed
US-20250304727-A1 PHOTOINITIATOR PACKAGE COMPRISING PHOSPHINE OXIDE PHOTOINITIATORS, COUMARIN-BASED SENSITIZERS AND AMINE ADDITIVES IGM GROUP B.V. (NL) 2025-10-02 US claimed
CN-120192293-A Organic luminescent material, preparation method of organic luminescent material and luminescent device 安徽省东超科技有限公司 2025-06-24 CN claimed
CN-120165029-A All-solid-state lithium metal battery and preparation method thereof 中国科学院上海高等研究院 2025-06-17 CN claimed
CN-120081814-A Organic light-emitting material, preparation method thereof and organic light-emitting device 安徽省东超科技有限公司 2025-06-03 CN claimed
WO-2025062323-A1 ENZYME LINKED IMMUNOASSAY WITH DIFFUSION RATE LIMITING MEDIUM ELLEON BIOTECH LIMITED (CN) 2025-03-27 WO claimed
EP-4519376-A1 PHOTOINITIATOR PACKAGE COMPRISING PHOSPHINE OXIDE PHOTOINITIATORS, COUMARIN-BASED SENSITIZERS AND AMINE ADDITIVES IGM Group B.V. (NL) 2025-03-12 EP claimed
US-4536322-A Fluorescent corrosive fluoride solution UNION CARBIDE CORPORATION (US) 1985-08-20 US claimed
EP-0140347-A2 Fluorescent corrosive fluoride solution UNION CARBIDE CORPORATION (US) 1985-05-08 EP claimed
US-4409140-A Substrates and method for determining enzymes SMITH ROBERT E (US) 1983-10-11 US claimed
EP-0034586-B1 4-TRIFLUOROMETHYLCOUMARIN PEPTIDE DERIVATIVES AND THEIR USE IN PROTEINASE ASSAYS Smith, Robert Eugene (US) 1983-08-31 EP claimed
EP-0018112-B1 SUBSTRATES AND METHOD FOR DETERMINING PROTEOLYTIC ENZYMES Smith, Robert Eugene (US) 1983-07-20 EP claimed
US-4294923-A AMINO ACID DERIVATIVE OF 7-AMINO-4-TRIFLUOROMETHYL COUMARIN HYDROLYZED TO FREE CHROMOPHORE SMITH ROBERT E 1981-10-13 US claimed
EP-0034586-A1 4-TRIFLUOROMETHYLCOUMARIN PEPTIDE DERIVATIVES AND THEIR USE IN PROTEINASE ASSAYS. SMITH ROBERT EUGENE (US) 1981-09-02 EP claimed
EP-0034586-A4 4-TRIFLUOROMETHYLCOUMARIN PEPTIDE DERIVATIVES AND THEIR USE IN PROTEINASE ASSAYS. SMITH ROBERT EUGENE (US) 1981-05-15 EP claimed
WO-1980002295-A1 4-TRIFLUOROMETHYLCOUMARIN PEPTIDE DERIVATIVES AND THEIR USE IN PROTEINASE ASSAYS SMITH R (US) 1980-10-30 WO claimed
EP-0018112-A1 Substrates and method for determining proteolytic enzymes Smith, Robert Eugene (US) 1980-10-29 EP claimed