SCHEMBL7973305

SCHEMBL7973305

Nc1cc(C(F)(F)F)c2ccc(=O)oc2c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.77
ALDH1A1 P00352 2/20 0.77
GAA P10253 2/20 0.77
HPGD P15428 2/20 0.77
CASP1 P29466 2/20 0.77
CASP7 P55210 2/20 0.77
HSD17B10 Q99714 2/20 0.77
MEN1 O00255 1/20 0.77
SRC P12931 1/20 0.77
KMT2A Q03164 1/20 0.77
ATM Q13315 1/20 0.77
NPSR1 Q6W5P4 1/20 0.77
TLR9 Q9NR96 1/20 0.77
HSD17B3 P37058 1/20 0.58
AR P10275 12/20 0.51
MAP2K1 Q02750 1/20 0.49
MCL1 Q07820 1/20 0.49
AGER Q15109 2/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL144309 0.87 KDM4E (1.00) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL29356441 0.87 KDM4E (1.00) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL15843573 0.81 HSD17B3 (0.59) KDM4EALDH1A1GAAHPGDCASP1
Glycine SCHEMBL9259892 0.77 KDM4E (0.79) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL8629120 0.77 NQO1 (0.55) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL30124129 0.77 NQO1 (0.55) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL4620259 0.76 KDM4E (0.68) KDM4EALDH1A1GAAHPGDCASP1
Alanine SCHEMBL15556780 0.75 KDM4E (0.75) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL15842662 0.75 HSD17B3 (0.69) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL2169023 0.74 ALDH1A1 (0.74) KDM4EALDH1A1GAAHPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6277583-B1 COMBINING A MIXTURE OF PROTEINS COMPRISING THE TARGET PROTEIN WITH AN AFFINITY LABEL CONJUGATE COMPRISING AN OLIGOMER AND A BIOLOGICALLY ACTIVE COMPOUND AND HAS AN ACTIVATED FUNCTIONAL GROUP WHICH COVALENTLY BONDS TO THE TARGET PROTEIN CONJUCHEM, INC. (CA) 2001-08-21 US disclosed
EP-0885390-A1 AFFINITY LABELING LIBRARIES AND APPLICATIONS THEREOF Redcell Canada Inc. (CA) 1998-12-23 EP disclosed
WO-1997029372-A1 AFFINITY LABELING LIBRARIES AND APPLICATIONS THEREOF CONJUCHEM, INC. (CA) 1997-08-14 WO disclosed