SCHEMBL14432255

SCHEMBL14432255

CNCCOC(=O)c1cc(C(=O)N2CC[C@H](C)Nc3ccccc32)ccc1-c1ccc2[nH]ccc2c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.36
OXTR P30559 1/20 0.35
GHSR Q92847 10/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
MAP3K11 Q16584 1/20 0.33
XIAP P98170 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4912744 0.91 MAPK14 (0.38) MAPK14OXTRGHSRGPBAR1
SCHEMBL14432384 0.90 CTSK (0.34) MAPK14OXTRGHSRGPBAR1
SCHEMBL14258886 0.90 KDR (0.39) MAPK14OXTRGHSRGPBAR1
SCHEMBL4909403 0.90 MAPK14 (0.36) MAPK14OXTRGHSRGPBAR1
SCHEMBL4933816 0.89 MAPK14 (0.37) MAPK14OXTRGHSRGPBAR1
SCHEMBL4933826 0.89 MAPK14 (0.37) MAPK14OXTRGHSRGPBAR1
SCHEMBL4910784 0.89 HRH3 (0.39) MAPK14OXTRGHSRGPBAR1MAP3K11
SCHEMBL14258848 0.89 OXTR (0.36) MAPK14OXTRGHSRGPBAR1
SCHEMBL4908666 0.88 OXTR (0.35) MAPK14OXTRGHSRGPBAR1
SCHEMBL4914320 0.88 ALDH1A1 (0.37) MAPK14OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1820799-A1 2,3,4,5-TETRAHYDRO-1H-1,5-BENZODIAZEPINE DERIVATIVE AND MEDICINAL COMPOSITION Wakamoto Pharmaceutical Co., Ltd. (JP) 2007-08-22 EP disclosed