SCHEMBL14435758

SCHEMBL14435758

CC(=O)c1cc(Br)ccc1N=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.46
MAOA P21397 1/20 0.46
CES2 O00748 1/20 0.42
GALR3 O60755 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GLA P06280 1/20 0.40
PLAU P00749 1/20 0.39
MAPT P10636 3/20 0.38
POLB P06746 2/20 0.38
MAPK1 P28482 1/20 0.38
GAA P10253 1/20 0.38
GSTA1 P08263 3/20 0.38
MYC P01106 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28238985 0.82 KDM4E (0.55) CES2GALR3CYP1A2CYP2C9HPGD
SCHEMBL13952292 0.78 CSNK2A1 (0.42) HPGDALDH1A1KDM4EMAPTPOLB
SCHEMBL30864269 0.77 MAOA (0.53) PTGDR2MAOACES2GALR3CYP1A2
SCHEMBL28237983 0.76 ALDH1A1 (0.50) HPGDALDH1A1MAPTMAPK1GAA
SCHEMBL25843039 0.76 MAOA (0.45) PTGDR2MAOACES2GALR3CYP1A2
SCHEMBL1310573 0.75 MAPT (0.51) PTGDR2MAOACES2GALR3CYP1A2
SCHEMBL2507576 0.75 MAOA (0.51) PTGDR2MAOACES2GALR3CYP1A2
SCHEMBL13498242 0.74 CYP4F2 (0.39) MAOAKDM4ECA12CA9
SCHEMBL6054167 0.74 ALDH1A1 (0.56) CYP1A2CYP2C9HPGDCYP2C19ALDH1A1
SCHEMBL309016 0.74 HPGD (0.69) PTGDR2MAOACES2GALR3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324032-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2014-10-01 EP disclosed
WO-2007088462-A1 SPIROCHROMANE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-08-09 WO disclosed