SCHEMBL14437486

SCHEMBL14437486

NC(=O)C(c1ccccc1)(c1ccccc1)c1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 15/20 0.65
KCNE1 P15382 1/20 0.54
KCNQ1 P51787 1/20 0.54
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.38
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL812971 0.81 KCNN4 (0.76) KCNN4KCNE1KCNQ1MAPTKMT2A
SCHEMBL13427553 0.81 KCNN4 (0.46) KCNN4KCNE1KCNQ1MAPTKMT2A
SCHEMBL2337394 0.78 KCNN4 (1.00) KCNN4KCNE1KCNQ1MAPTKMT2A
Senicapoc SCHEMBL1443805 0.78 KCNN4 (1.00) KCNN4KCNE1KCNQ1MAPTKMT2A
SCHEMBL1784375 0.76 KCNN4 (1.00) KCNN4KCNE1KCNQ1MAPTKMT2A
SCHEMBL2332073 0.76 KCNN4 (1.00) KCNN4KCNE1KCNQ1MAPTKMT2A
SCHEMBL18782553 0.74 KCNN4 (0.72) KCNN4KCNE1KCNQ1MAPTKMT2A
SCHEMBL13950934 0.74 KCNN4 (1.00) KCNN4KCNE1KCNQ1MAPTKMT2A
SCHEMBL3526866 0.74 KCNN4 (0.56) KCNN4KCNE1KCNQ1MAPTKMT2A
SCHEMBL14437487 0.73 KCNN4 (1.00) KCNN4KCNE1KCNQ1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180042872-A1 METHODS FOR TREATING MALARIA USING POTASSIUM CHANNEL INHIBITORS THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2018-02-15 US disclosed
WO-2017070536-A1 METHODS AND AGENTS FOR TREATING DISEASES ANGION BIOMEDICA CORP. (US) 2017-04-27 WO disclosed
US-20070185209-A1 Treatment methods using triaryl methane compounds ICAGEN, INC. (US) 2007-08-09 US disclosed
US-20070185209-A1 Treatment methods using triaryl methane compounds ICAGEN, INC. (US) 2007-08-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185209-A1 Treatment methods using triaryl methane compounds KCNH3, KCNH2, KCNJ2 KCNN4 37/4885KCNE1 20/4885KCNQ1 23/4885
US-20180042872-A1 METHODS FOR TREATING MALARIA USING POTASSIUM CHANNEL INHIBITORS KCNN1, KCNN2, KCNN3 KCNN4 10/4885KCNE1 41/4885KCNQ1 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.