Gw786460X

Gw786460X

SCHEMBL144632

Cc1cccc(-c2n[nH]cc2-c2ccc3ncccc3n2)n1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 20/20 0.60
MAPK14 Q16539 3/20 0.46
MTOR P42345 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gw786460X SCHEMBL29398528 1.00 TGFBR1 (0.60) TGFBR1MAPK14MTOR
Gw786460X SCHEMBL29889251 0.99 TGFBR1 (0.59) TGFBR1MAPK14MTOR
Gw786460X SCHEMBL26962436 0.99 TGFBR1 (0.59) TGFBR1MAPK14MTOR
SCHEMBL20822412 0.86 TGFBR1 (0.44) TGFBR1MAPK14
SCHEMBL373397 0.84 TGFBR1 (0.56) TGFBR1MAPK14MTOR
SCHEMBL25822564 0.83 TGFBR1 (0.44) TGFBR1MAPK14MTOR
SCHEMBL27842262 0.82 TGFBR1 (0.41) TGFBR1MAPK14
SCHEMBL25085206 0.82 TGFBR1 (0.47) TGFBR1MAPK14MTOR
SCHEMBL30156338 0.82 TGFBR1 (0.47) TGFBR1MAPK14MTOR
Hydrochloric Acid SCHEMBL31572311 0.82 AR (0.50) TGFBR1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1110 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260097083-A1 METHOD FOR PRODUCING PANCREATIC ENDODERM CELLS KYOTO UNIVERSITY (JP) 2026-04-09 US claimed
EP-4692329-A1 COMPOSITION FOR INDUCING DIRECT DIFFERENTIATION OF STEM CELLS INTO CORNEAL ENDOTHELIAL CELLS AND METHOD FOR INDUCING DIRECT DIFFERENTIATION USING SAME The Asan Foundation (KR) 2026-02-11 EP claimed
EP-3784232-B1 IMPROVED METHODS FOR INDUCING TISSUE REGENERATION AND SENOLYSIS IN MAMMALIAN CELLS AGEX THERAPEUTICS INC (US) 2026-02-11 EP claimed
US-12427147-B2 Retinal ganglion cell death inhibitor SENJU PHARMACEUTICAL CO., LTD. (JP) 2025-09-30 US claimed
EP-3047017-B1 METHODS OF MAMMALIAN RETINAL STEM CELL PRODUCTION AND APPLICATIONS UNIV CALIFORNIA (US) 2025-09-10 EP claimed
EP-4596675-A1 METHOD FOR PRODUCING PANCREATIC ENDODERM CELLS Kyoto University (JP) 2025-08-06 EP claimed
US-12371664-B2 Medium for direct differentiation of pluripotent stem cell-derived mesenchymal stem cell, method for preparing mesenchymal stem cell by using same, and mesenchymal stem cell prepared thereby CHA BIOTECH CO., LTD. (KR) 2025-07-29 US claimed
US-20250188420-A1 MATURING AGENT HAVING BOTH OF ALK5 INHIBITORY ACTIVITY AND CDK8/19 INHIBITORY ACTIVITY Orizuru Therapeutics, Inc. (JP) 2025-06-12 US claimed
EP-4516894-A1 MATURING AGENT HAVING BOTH OF ALK5 INHIBITORY ACTIVITY AND CDK8/19 INHIBITORY ACTIVITY Orizuru Therapeutics, Inc. (JP) 2025-03-05 EP claimed
US-RE50313-E1 Musculoskeletal stem cell and medium for inducing differentiation of musculoskeletal stem cell CELLATOZ THERAPEUTICS, INC. (KR) 2025-02-25 US claimed
US-20130236436-A1 EXPANDABLE CELL SOURCE OF NEURONAL STEM CELL POPULATIONS AND METHODS FOR OBTAINING AND USNIG THEM ZHANG KANG (US) 2013-09-12 US claimed
US-20130071931-A1 PROCESS FOR HEPATIC DIFFERENTIATION FROM INDUCED HEPATIC STEM CELLS, AND INDUCED HEPATIC PROGENITOR CELLS DIFFERENTIATED THEREBY NATIONAL CANCER CENTER (JP) 2013-03-21 US claimed
US-20130022986-A1 METHOD FOR MANUFACTURING PANCREATIC-HORMONE-PRODUCING CELLS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-01-24 US claimed
US-8298825-B1 TGF-beta receptor inhibitors to enhance direct reprogramming THE GENERAL HOSPITAL CORPORATION (US) 2012-10-30 US claimed
EP-2505639-A1 METHOD FOR MANUFACTURING PANCREATIC-HORMONE-PRODUCING CELLS Takeda Pharmaceutical Company Limited (JP) 2012-10-03 EP claimed
EP-2229434-B1 DIFFERENTIATION OF HUMAN EMBRYONIC STEM CELLS LIFESCAN INC (US) 2011-09-07 EP claimed
EP-2229434-A2 DIFFERENTIATION OF HUMAN EMBRYONIC STEM CELLS Lifescan, Inc. (US) 2010-09-22 EP claimed
US-20100167300-A1 MICROENVIRONMENT NICHE ASSAY FOR CiPS SCREENING ESMAELI-AZAD, BABAK 2010-07-01 US claimed
US-20090170198-A1 Differentiation of human embryonic stem cells JANSSEN BIOTECH, INC. 2009-07-02 US claimed
WO-2009070592-A2 DIFFERENTIATION OF HUMAN EMBRYONIC STEM CELLS LIFESCAN, INC. (US) 2009-06-04 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260097083-A1 METHOD FOR PRODUCING PANCREATIC ENDODERM CELLS PNLIP, GIPR, CEL TGFBR1 1634/4885MAPK14 580/4885MTOR 769/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.