SCHEMBL1448490

SCHEMBL1448490

O=C1c2ccccc2C(=O)N1CCCCCCCCCO

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.70
ALDH1A1 P00352 2/20 0.70
MEN1 O00255 2/20 0.70
KMT2A Q03164 2/20 0.70
SMN1; SMN2 Q16637 2/20 0.70
RGS12 O14924 1/20 0.70
NPC1 O15118 1/20 0.70
LMNA P02545 1/20 0.70
PABPC1 P11940 1/20 0.70
HTT P42858 1/20 0.70
RECQL P46063 1/20 0.70
RAB9A P51151 1/20 0.70
TDP1 Q9NUW8 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.64
HDAC8 Q9BY41 3/20 0.61
HDAC3 O15379 2/20 0.61
HDAC4 P56524 2/20 0.61
HDAC1 Q13547 2/20 0.61
HDAC7 Q8WUI4 2/20 0.61
HDAC2 Q92769 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3468337 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7544499 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7352888 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7285741 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7296911 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL4179085 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL17275126 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL1162502 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL3468673 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL1703575 1.00 KDM4E (0.70) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0662834-A4 NOVEL EPOXIDE-CONTAINING COMPOUNDS. CELL THERAPEUTICS INC (US) 1996-04-17 EP claimed
EP-0662834-A1 NOVEL EPOXIDE-CONTAINING COMPOUNDS CELL THERAPEUTICS, INC. (US) 1995-07-19 EP claimed
WO-1994006431-A1 NOVEL EPOXIDE-CONTAINING COMPOUNDS CELL THERAPEUTICS, INC. (US) 1994-03-31 WO claimed
US-12624044-B2 SMARCA degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2026-05-12 US disclosed
CN-118255685-A Tricyclic compound, pharmaceutical composition and application thereof 珂阑(上海)医药科技有限公司 2024-06-28 CN disclosed
US-11833208-B2 PLK1 selective degradation inducing compound UPPTHERA, INC. (KR) 2023-12-05 US disclosed
US-20230372498-A1 PLK1 SELECTIVE DEGRADATION INDUCING COMPOUND UPPTHERA (KR) 2023-11-23 US disclosed
US-20230348362-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS Suzhou Abogen Biosciences Co., Ltd. (CN) 2023-11-02 US disclosed
US-20230348362-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS Suzhou Abogen Biosciences Co., Ltd. (CN) 2023-11-02 US disclosed
CN-116444494-A Compound for targeted degradation of BUB1B and BUB1 protein, and preparation method and application thereof 浙江大学 2023-07-18 CN disclosed
US-20230072658-A1 SMARCA DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2023-03-09 US disclosed
EP-1755684-A2 ALBUMIN-BINDING CONJUGATES COMPRISING A FATTY ACID AND PEG Celltech R&D Limited (GB) 2007-02-28 EP disclosed
WO-2005117984-A2 ALBUMIN-BINDING CONJUGATES COMPRISING A FATTY ACID AND PEG CELLTECH R & D LIMITED (GB) 2005-12-15 WO disclosed
WO-2002016314-A1 SUBSTITUTED POLYAMINE COMPOUNDS H. LUNDBECK A/S (DK) 2002-02-28 WO disclosed
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230372498-A1 PLK1 SELECTIVE DEGRADATION INDUCING COMPOUND PLK1, BUB1B, BUB1 KDM4E 1207/4885ALDH1A1 3592/4885MEN1 1845/4885
US-20230348362-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS CETP, NPC1, LCAT KDM4E 3784/4885ALDH1A1 4264/4885MEN1 1909/4885
US-12624044-B2 SMARCA degraders and uses thereof SMARCA1, SMARCC1, SMARCA2 KDM4E 315/4885ALDH1A1 3543/4885MEN1 1936/4885
US-11833208-B2 PLK1 selective degradation inducing compound PLK1, BUB1B, BUB1 KDM4E 1207/4885ALDH1A1 3592/4885MEN1 1845/4885
US-20230072658-A1 SMARCA DEGRADERS AND USES THEREOF SMARCA1, SMARCB1, SMARCE1 KDM4E 624/4885ALDH1A1 3736/4885MEN1 1348/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.