SCHEMBL14503530

SCHEMBL14503530

Cc1ccnc(NS(=O)(=O)c2ccc(Nc3nc(N4CCCCC4)nc(N4CCCCC4)n3)cc2)n1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.58
ALDH1A1 P00352 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.56
FASN P49327 1/20 0.56
MAPT P10636 1/20 0.54
CYP2C9 P11712 1/20 0.54
NPSR1 Q6W5P4 2/20 0.53
KMT2A Q03164 1/20 0.53
POLB P06746 1/20 0.53
PTGS2 P35354 2/20 0.51
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5401247 0.84 MAPK1 (0.54) MAPK1ALDH1A1FASNMAPTCYP2C9
SCHEMBL14503148 0.80 MAPT (0.55) MAPK1ALDH1A1MAPTNPSR1KMT2A
SCHEMBL14503062 0.80 NPSR1 (0.56) MAPK1ALDH1A1SMN1; SMN2MAPTCYP2C9
SCHEMBL14503557 0.78 PTGS2 (0.50) ALDH1A1SMN1; SMN2MAPTCYP2C9NPSR1
SCHEMBL14503065 0.77 EDNRA (0.55) CYP2C9KMT2A
SCHEMBL14504503 0.76 NPSR1 (0.68) ALDH1A1SMN1; SMN2MAPTNPSR1KMT2A
SCHEMBL14503056 0.75 CA1 (0.76) MAPTNPSR1KMT2APTGS2LMNA
SCHEMBL14503488 0.74 ESR1 (0.60) ALDH1A1NPSR1KMT2APTGS2LMNA
SCHEMBL14081433 0.73 MAPT (0.78) MAPK1ALDH1A1FASNMAPTCYP2C9
SCHEMBL14503936 0.73 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2MAPTCYP2C9NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7223759-B2 Antibacterial 3,5-diaminopiperidine-substituted aromatic and heteroaromatic compounds ANADYS PHARMACEUTICALS, INC. (US) 2007-05-29 US disclosed
US-7223759-B2 Antibacterial 3,5-diaminopiperidine-substituted aromatic and heteroaromatic compounds ANADYS PHARMACEUTICALS, INC. (US) 2007-05-29 US disclosed