SCHEMBL14507697

SCHEMBL14507697

CCCn1cc(C(N)=O)ccc1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.45
NPC1 O15118 3/20 0.43
MAP2K2 P36507 1/20 0.41
MAP2K1 Q02750 1/20 0.41
BRD4 O60885 4/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
BRD2 P25440 1/20 0.40
BRD3 Q15059 1/20 0.40
BRDT Q58F21 1/20 0.40
BRPF1 P55201 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PARP10 Q53GL7 1/20 0.40
BRD9 Q9H8M2 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
LMNA P02545 1/20 0.38
EPHX2 P34913 2/20 0.38
FABP6 P51161 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27774707 0.90 TLR8 (0.52) TLR8NPC1BRD4KDM4EALDH1A1
SCHEMBL23805183 0.86 KDM4E (0.42) TLR8NPC1MAP2K2MAP2K1BRD4
SCHEMBL3161296 0.84 L3MBTL1 (0.45) BRD4KDM4EALDH1A1BRD2BRD3
SCHEMBL14507440 0.83 EPHX2 (0.56) TLR8MAP2K2MAP2K1BRD4KDM4E
SCHEMBL6496861 0.81 TLR8 (0.41) TLR8MAP2K2MAP2K1BRD4KDM4E
SCHEMBL21395223 0.80 LMNA (0.59) TLR8BRD4KDM4EALDH1A1BRD2
SCHEMBL14507698 0.80 ALDH1A1 (0.36) TLR8NPC1BRD4KDM4EALDH1A1
SCHEMBL12095050 0.79 KDM4E (0.43) TLR8BRD4KDM4EALDH1A1BRD2
SCHEMBL13701807 0.76 BRD4 (0.45) BRD4ALDH1A1BRD2BRD3BRDT
SCHEMBL13039896 0.76 LMNA (0.43) BRD4KDM4EALDH1A1BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007067836-A2 SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-06-14 WO disclosed