SCHEMBL14516263

SCHEMBL14516263

CCCCNc1nccc(OC)n1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.52
MERTK Q12866 2/20 0.48
DNM2 P50570 2/20 0.48
TLR8 Q9NR97 1/20 0.46
MAPK8 P45983 1/20 0.45
CCR4 P51679 4/20 0.44
PDPK1 O15530 6/20 0.43
FLT3 P36888 1/20 0.42
TYRO3 Q06418 1/20 0.42
GAS6 Q14393 1/20 0.42
GBA1 P04062 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14516259 0.90 CYP1A2 (0.45) HRH4MERTKDNM2CCR4PDPK1
SCHEMBL12280402 0.83 DYRK1B (0.46) HRH4DNM2CCR4PDPK1
SCHEMBL28860465 0.83 MKNK1 (0.42) CCR4PDPK1
SCHEMBL28020340 0.82 MKNK1 (0.50) CCR4PDPK1
SCHEMBL8439579 0.80 GBA1 (0.46) DNM2TLR8GBA1
SCHEMBL19788436 0.79 PDPK1 (0.48) HRH4DNM2CCR4PDPK1
SCHEMBL10055017 0.78 CLK4 (0.52)
SCHEMBL19477219 0.78 DNM2 (0.71) HRH4MERTKDNM2TLR8MAPK8
SCHEMBL13403107 0.78 HRH4 (0.56) HRH4MERTKDNM2TLR8MAPK8
SCHEMBL14619914 0.77 HRH4 (0.55) HRH4MERTKDNM2TLR8MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230346951-A1 MOLECULAR DEGRADERS OF EXTRACELLULAR PROTEINS YALE UNIVERSITY 2023-11-02 US disclosed
US-7205410-B2 4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders JANSSEN PHARMACEUTICA, N.V. (BE) 2007-04-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230346951-A1 MOLECULAR DEGRADERS OF EXTRACELLULAR PROTEINS ASGR1, MSR1, LDLR HRH4 3145/4885MERTK 1284/4885DNM2 3515/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.