Irloxacin

Irloxacin

SCHEMBL145215

CCn1cc(C(=O)O)c(=O)c2cc(F)c(-n3cccc3)cc21

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 1/20 0.67
KDM4E B2RXH2 7/20 0.66
HPGD P15428 5/20 0.66
ALDH1A1 P00352 5/20 0.66
HSD17B10 Q99714 4/20 0.66
HTT P42858 4/20 0.66
LMNA P02545 3/20 0.66
TSHR P16473 2/20 0.66
BRD4 O60885 1/20 0.66
CYP2J2 P51589 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66
MEN1 O00255 5/20 0.61
KMT2A Q03164 5/20 0.61
NPC1 O15118 1/20 0.61
USP2 O75604 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
HIF1A Q16665 1/20 0.57
POLB P06746 1/20 0.57
TAAR1 Q96RJ0 1/20 0.57
PIK3CG P48736 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Irloxacin SCHEMBL9743690 0.99 DRD3 (0.66) DRD3KDM4EHPGDALDH1A1HSD17B10
Irloxacin SCHEMBL9743701 0.99 DRD3 (0.66) DRD3KDM4EHPGDALDH1A1HSD17B10
SCHEMBL10671111 0.91 ALDH1A1 (0.59) DRD3KDM4EHPGDALDH1A1HSD17B10
SCHEMBL16518634 0.89 DRD3 (0.54) DRD3KDM4EHPGDALDH1A1HSD17B10
Irloxacin SCHEMBL9743694 0.88 DRD3 (0.53) DRD3KDM4EHPGDALDH1A1HSD17B10
SCHEMBL10372171 0.88 ALDH1A1 (0.67) DRD3KDM4EHPGDALDH1A1HSD17B10
SCHEMBL9757197 0.87 DRD3 (0.64) DRD3KDM4EHPGDALDH1A1HSD17B10
SCHEMBL10369898 0.87 ALDH1A1 (0.57) DRD3KDM4EHPGDALDH1A1HSD17B10
SCHEMBL10972617 0.86 KDM4E (0.68) DRD3KDM4EHPGDALDH1A1HSD17B10
SCHEMBL9700859 0.85 DRD3 (0.61) DRD3KDM4EHPGDALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1176 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118354776-A Methods and compositions for enhanced efficacy and reduced toxicity of non-implanted CD8 depleted allogeneic donor lymphocyte infusions 约翰霍普金斯大学 2024-07-16 CN claimed
US-20230285572-A1 TARGETED DELIVERY OF THERAPEUTIC AGENTS SEPELO THERAPEUTICS, LLC 2023-09-14 US claimed
EP-4188433-A2 TARGETED DELIVERY OF THERAPEUTIC AGENTS Sepelo Therapeutics, LLC (US) 2023-06-07 EP claimed
WO-2023028364-A1 TARGETED COMPOSITIONS AND USES THEROF SEPELO THERAPEUTICS, LLC (US) 2023-03-02 WO claimed
WO-2022031761-A2 TARGETED DELIVERY OF THERAPEUTIC AGENTS SEPELO THERAPEUTICS, LLC (US) 2022-02-10 WO claimed
US-10953073-B2 XTEN conjugate compositions and methods of making same AMUNIX PHARMACEUTICALS, INC. (US) 2021-03-23 US claimed
CN-111135182-A Antibacterial product and preparation method and application thereof 心远(广州)药物研究有限公司 2020-05-12 CN claimed
CN-109847109-A A kind of contact lens carrying medicine 滕宇池 2019-06-07 CN claimed
US-20190099363-A1 CHEMICALLY MODIFIED SMALL MOLECULES REDHILL BIOPHARMA LTD. (IL) 2019-04-04 US claimed
CN-104725628-B A kind of single functionalization branched polyethylene glycol, preparation method and its bio-related substance containing degradable group 厦门赛诺邦格生物科技股份有限公司 2018-04-17 CN claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
CN-1500488-A Oral colon-positioned medicine composition for curing bacillary dysentery 北京东方凯恩医药科技有限公司 2004-06-02 CN claimed
US-4895803-A QUINOLINE-OR NAPHTHAPYRIDINE/1,8-/ DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1990-01-23 US claimed
US-4853225-A Process for implanting a medicament depot MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1989-08-01 US claimed
US-4844902-A Topically applicable formulations of gyrase inhibitors in combination with corticosteroids BAYER AKTIENGESELLSCHAFT (DE) 1989-07-04 US claimed
EP-0280915-A2 Preparations for topical use of gyrase inhibitors in combination with corticosteroids BAYER AG (DE) 1988-09-07 EP claimed
EP-0134165-B1 7-(PYRROL-1-YL)-1-ETHYL-1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXYLIC ACID AND 7-(PYRROL-1-YL)-1-ETHYL-1,4-DIHYDRO-4-OXO-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS PROVESAN S.A. (CH) 1988-06-08 EP claimed
US-4552882-A 7-(1-Pyrrolyl) derivatives of 1-ethyl-1,4-dihydro-4-oxoquinoline-3-carboxylic acids and 1-ethyl-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acids and their use as antimicrobial agents PROVESAN, SA (CH) 1985-11-12 US claimed
EP-0155244-A2 1-Ethyl-6-fluoro-7-(1H-pirrol-1-yl)-1,4-dihydro-4-oxoquinoline-3-carboxylic acid: preparation and antimicrobial activities BIOCHEM DESIGN S.r.l. (IT) 1985-09-18 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10953073-B2 XTEN conjugate compositions and methods of making same XPA, TXLNA, NGLY1 DRD3 2834/4885KDM4E 2338/4885HPGD 2116/4885
US-20190099363-A1 CHEMICALLY MODIFIED SMALL MOLECULES H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CD44, ELANE DRD3 2250/4885KDM4E 2294/4885HPGD 678/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.