SCHEMBL14539263

SCHEMBL14539263

C=C(c1ccc(F)cc1)N(C)C(C)=O

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
BCL2L1 Q07817 1/20 0.39
BAD Q92934 1/20 0.39
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
PTPN1 P18031 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
APP P05067 1/20 0.38
HTR7 P34969 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14539265 0.84 MAPT (0.43) NPC1RAB9AMAPT
SCHEMBL14539266 0.80 EGFR (0.47) CES2CES1NPC1RAB9AMAPT
SCHEMBL31301102 0.78 HDAC1 (0.47) NPC1RAB9AMAPT
SCHEMBL9266647 0.77 MAOA (0.49) CES2CES1CYP1A2CYP2C19CA1
SCHEMBL29156800 0.74 KMT2A (0.42) CES2CES1CYP1A2CYP2C19CA1
SCHEMBL38650903 0.73 NR3C2 (0.44) NPC1RAB9AMAPT
SCHEMBL27720360 0.71 CES2 (0.52) CES2CES1CYP1A2CYP2C19CA1
SCHEMBL27919033 0.71 BCL2L1 (0.68) CES2CES1CA1CA2BCL2L1
SCHEMBL11802097 0.71 CES2 (0.65) CES2CES1CYP1A2CYP2C19CA1
SCHEMBL29083762 0.71 TAS2R14 (0.49) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007057658-A1 PALLADIUM CATALYSED HECK ARYLATION OR VINYLATION OF 1-SUBSTITUTED OLEFINS THE UNIVERSITY OF LIVERPOOL (GB) 2007-05-24 WO disclosed