SCHEMBL14569802

SCHEMBL14569802

CC1C(c2ccccc2)N(C)C(=O)N1C

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.72
MEN1 O00255 3/20 0.72
TSHR P16473 3/20 0.72
ALDH1A1 P00352 3/20 0.45
ATM Q13315 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
PABPC1 P11940 1/20 0.42
BRD4 O60885 3/20 0.38
HTR1A P08908 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ELANE P08246 1/20 0.37
SRD5A1 P18405 1/20 0.36
ADRA2C P18825 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2733150 0.87 TSHR (0.65) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL2733147 0.87 TSHR (0.65) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL418149 0.80 KMT2A (0.54) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL463912 0.79 TSHR (0.56) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL416900 0.76 TSHR (0.52) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL464236 0.76 MEN1 (0.52) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL7806213 0.74 TSHR (0.51) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL13557184 0.73 KMT2A (0.50) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL8517882 0.73 ATM (0.48) KMT2AMEN1TSHRALDH1A1ATM
SCHEMBL30561555 0.73 ATM (0.48) KMT2AMEN1TSHRALDH1A1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7196081-B2 Compounds with hydroxycarbonyl-halogenoalkyl side chains CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2007-03-27 US disclosed