SCHEMBL1457110

SCHEMBL1457110

S=C=NCCCc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MIF P14174 6/20 1.00
NAAA Q02083 7/20 0.85
TRPA1 O75762 2/20 0.77
CYP2E1 P05181 1/20 0.77
CYP2A6 P11509 1/20 0.77
HIF1A Q16665 1/20 0.77
CYP2A13 Q16696 1/20 0.77
EPAS1 Q99814 1/20 0.77
ALDH1A1 P00352 1/20 0.57
CYP3A4 P08684 1/20 0.57
HPGD P15428 1/20 0.57
HTR3A P46098 1/20 0.57
KEAP1 Q14145 5/20 0.56
NFE2L2 Q16236 5/20 0.56
MAOA P21397 1/20 0.54
MAOB P27338 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenylbutyl Isothiocyanate SCHEMBL1526828 0.94 MIF (1.00) MIFNAAATRPA1CYP2E1CYP2A6
SCHEMBL17274357 0.92 NAAA (1.00) MIFNAAATRPA1CYP2E1CYP2A6
SCHEMBL17274355 0.92 NAAA (1.00) MIFNAAATRPA1CYP2E1CYP2A6
SCHEMBL17274466 0.92 NAAA (1.00) MIFNAAATRPA1CYP2E1CYP2A6
Phenylhexyl Isothiocyanate SCHEMBL7809 0.92 NAAA (1.00) MIFNAAATRPA1CYP2E1CYP2A6
SCHEMBL17274428 0.92 NAAA (1.00) MIFNAAATRPA1CYP2E1CYP2A6
SCHEMBL9493211 0.92 NAAA (1.00) MIFNAAATRPA1CYP2E1CYP2A6
SCHEMBL331147 0.89 MIF (0.80) MIFNAAATRPA1CYP2E1CYP2A6
Phenethylisothiocyanate SCHEMBL156960 0.87 MIF (1.00) MIFNAAATRPA1CYP2E1CYP2A6
Phenethylisothiocyanate SCHEMBL27616786 0.87 MIF (1.00) MIFNAAATRPA1CYP2E1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 150 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118873488-A Coacervate and method for the production and use thereof 海诺生物科技有限公司 2024-11-01 CN claimed
CN-115429785-A Composition for improving bioavailability and treatment effect of isothiocyanate compounds 无锡杰西医药股份有限公司 2022-12-06 CN claimed
EP-3681476-B1 TRANSDERMAL FORMULATIONS TYME INC (US) 2022-09-14 EP claimed
CN-104173272-B Sustained-release preparation of isothiocyanate compounds 无锡杰西医药股份有限公司 2021-07-06 CN claimed
CN-104117064-B Combined application of isothiocyanate compounds and hormone drugs 无锡杰西医药股份有限公司 2021-02-26 CN claimed
US-20200405680-A1 TRANSDERMAL FORMULATIONS TYME, INC. (US) 2020-12-31 US claimed
EP-3034076-B1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE JC WUXI COMPANY INC (CN) 2020-09-30 EP claimed
EP-3681476-A1 TRANSDERMAL FORMULATIONS Tyme, Inc. (US) 2020-07-22 EP claimed
CN-111328278-A Transdermal preparation 迪美公司 2020-06-23 CN claimed
CN-110041522-B Polyethylene glycol-polylysine/isothiocyanate bonding substance and application thereof as drug carrier 浙江大学 2020-05-29 CN claimed
WO-2019055747-A1 TRANSDERMAL FORMULATIONS TYME, INC. (US) 2019-03-21 WO claimed
US-10010520-B2 Combined application of isothiocyanate compound and anti-cancer medicine JC (WUXI) COMPANY, INC. (CN) 2018-07-03 US claimed
CN-106279529-A A kind of positive osmotic drive liquid for waste water process and preparation method thereof 中南林业科技大学 2017-01-04 CN claimed
US-20160250175-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE JC (WUXI) COMPANY, INC. (CN) 2016-09-01 US claimed
EP-3034076-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE JC (Wuxi) COMPANY, Inc. (CN) 2016-06-22 EP claimed
CN-104502478-B A kind of arginine assay method based on LC-MS/MS newly 3D BIOOPTIMA CO., LTD. (CN) 2016-03-30 CN claimed
CN-105267967-A Combined application of isothiocyanate-type compound and anti-cancer drug acting or affecting DNA WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2016-01-27 CN claimed
CN-104502478-A Novel arginine determination method based on LC-MS/MS 3D BIOOPTIMA CO LTD 2015-04-08 CN claimed
CN-104415332-A Combined application between isothiocyanate-type compound and kinase inhibitor medicine in treatment of cancer WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2015-03-18 CN claimed
CN-104117064-A Combined application of isothiocyanate compound and hormone medicine WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2014-10-29 CN claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160250175-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE CHUK, KIT, MKI67 MIF 986/4885NAAA 3936/4885TRPA1 2138/4885
US-10010520-B2 Combined application of isothiocyanate compound and anti-cancer medicine CHUK, KIT, MKI67 MIF 986/4885NAAA 3936/4885TRPA1 2138/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.