SCHEMBL14573161

SCHEMBL14573161

NCCCOc1ccc2nccc(NC(=O)C3CCN(CCc4nc5c(F)cccc5[nH]4)CC3)c2n1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 6/20 0.40
PARP1 P09874 1/20 0.39
KCNH2 Q12809 6/20 0.38
SLC2A1 P11166 1/20 0.37
TP53 P04637 1/20 0.35
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5766014 0.91 CHRM3 (0.41) SLC40A1KCNH2
SCHEMBL14573148 0.91 KCNH2 (0.47) SLC40A1KCNH2SLC2A1
SCHEMBL5657252 0.88 SLC40A1 (0.37) SLC40A1PARP1KCNH2SLC2A1DRD2
SCHEMBL5765657 0.81 KCNH2 (0.47) SLC40A1KCNH2SLC2A1
SCHEMBL6661601 0.77 KCNH2 (0.45) SLC40A1KCNH2SLC2A1
SCHEMBL5774180 0.77 KCNH2 (0.42) SLC40A1KCNH2SLC2A1
SCHEMBL5657093 0.73 CHRNA7 (0.47) SLC40A1PARP1DRD2
SCHEMBL5656451 0.70 KDM4E (0.53) SLC40A1
SCHEMBL6214270 0.69 KCNH2 (0.51) KCNH2
SCHEMBL14573150 0.69 KCNH2 (0.51) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7186730-B2 Bicyclic nitrogen-containing heterocyclic derivatives for use as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2007-03-06 US disclosed