SCHEMBL5765657

SCHEMBL5765657

COc1ccc2nccc(NC(=O)OC3CCN(CCc4nc5c(F)cccc5[nH]4)CC3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.47
SLC40A1 Q9NP59 3/20 0.40
SLC2A1 P11166 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5766014 0.91 CHRM3 (0.41) KCNH2SLC40A1
SCHEMBL14573148 0.90 KCNH2 (0.47) KCNH2SLC40A1SLC2A1
SCHEMBL5774180 0.89 KCNH2 (0.42) KCNH2SLC40A1SLC2A1
SCHEMBL6661601 0.81 KCNH2 (0.45) KCNH2SLC40A1SLC2A1
SCHEMBL14573161 0.81 SLC40A1 (0.40) KCNH2SLC40A1SLC2A1
SCHEMBL5764918 0.79 KCNH2 (0.45) KCNH2
SCHEMBL5657252 0.79 SLC40A1 (0.37) KCNH2SLC40A1SLC2A1
SCHEMBL5765881 0.77 KCNH2 (0.45) KCNH2
SCHEMBL5764847 0.77 KCNH2 (0.48) KCNH2
SCHEMBL5764517 0.76 KCNH2 (0.58) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392686-B1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2006-10-18 EP claimed